CAPECITABINE

85/100 · Critical

Manufactured by H2-Pharma, LLC

Severe Adverse Reactions Common with Capecitabine Use

174,965 FDA adverse event reports analyzed

Last updated: 2026-05-12

About CAPECITABINE

CAPECITABINE is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by H2-Pharma, LLC. Based on analysis of 174,965 FDA adverse event reports, CAPECITABINE has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for CAPECITABINE include DIARRHOEA, DEATH, NAUSEA, PALMAR-PLANTAR ERYTHRODYSAESTHESIA SYNDROME, FATIGUE. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for CAPECITABINE.

AI Safety Analysis

Capecitabine has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 174,965 adverse event reports for this medication, which is primarily manufactured by H2-Pharma, Llc.

The most commonly reported adverse events include Diarrhoea, Death, Nausea. Of classified reports, 82.2% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Severe adverse reactions such as death, disease progression, and sepsis are frequently reported.

Diarrhoea and nausea are the most common gastrointestinal side effects. Neutropenia and thrombocytopenia are significant hematological concerns.

Patients taking Capecitabine should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Capecitabine can cause severe hematological and gastrointestinal side effects, and patients should be monitored closely for signs of toxicity. Drug interactions, particularly with other cytotoxic agents, should be avoided. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Capecitabine received a safety concern score of 85/100 (high concern). This is based on a 82.2% serious event ratio across 88,887 classified reports. The score accounts for 174,965 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

DIARRHOEA13,395 reports
DEATH8,723 reports
NAUSEA8,248 reports
PALMAR PLANTAR ERYTHRODYSAESTHESIA SYNDROME6,536 reports
FATIGUE6,329 reports
VOMITING6,134 reports
DISEASE PROGRESSION5,958 reports
MALIGNANT NEOPLASM PROGRESSION3,820 reports
OFF LABEL USE3,672 reports
ASTHENIA3,322 reports
DECREASED APPETITE3,172 reports
NEUTROPENIA3,046 reports
NEUROPATHY PERIPHERAL2,768 reports
DEHYDRATION2,716 reports
DYSPNOEA2,617 reports
DRUG INEFFECTIVE2,558 reports
THROMBOCYTOPENIA2,441 reports
PYREXIA2,420 reports
ANAEMIA2,310 reports
RASH2,220 reports
ABDOMINAL PAIN2,212 reports
PAIN2,170 reports
STOMATITIS2,062 reports
WEIGHT DECREASED1,995 reports
MUCOSAL INFLAMMATION1,954 reports
CONSTIPATION1,862 reports
METASTASES TO LIVER1,801 reports
PAIN IN EXTREMITY1,743 reports
MALAISE1,741 reports
DIZZINESS1,592 reports
HEADACHE1,543 reports
PARAESTHESIA1,527 reports
ERYTHEMA1,455 reports
PNEUMONIA1,325 reports
NEOPLASM PROGRESSION1,294 reports
METASTASES TO BONE1,284 reports
PLATELET COUNT DECREASED1,257 reports
HYPOAESTHESIA1,238 reports
SEPSIS1,200 reports
BREAST CANCER METASTATIC1,188 reports
SKIN EXFOLIATION1,179 reports
FEBRILE NEUTROPENIA1,164 reports
GENERAL PHYSICAL HEALTH DETERIORATION1,156 reports
DRY SKIN1,150 reports
MYELOSUPPRESSION1,140 reports
WHITE BLOOD CELL COUNT DECREASED1,130 reports
ABDOMINAL PAIN UPPER1,125 reports
HYPERTENSION1,125 reports
CHEST PAIN1,109 reports
LEUKOPENIA1,102 reports
PULMONARY EMBOLISM1,078 reports
METASTASES TO CENTRAL NERVOUS SYSTEM1,049 reports
BACK PAIN1,033 reports
COUGH1,024 reports
TOXICITY TO VARIOUS AGENTS1,002 reports
METASTASES TO LUNG994 reports
HYPOKALAEMIA987 reports
ALOPECIA942 reports
BREAST CANCER937 reports
PLEURAL EFFUSION934 reports
FALL931 reports
INFECTION918 reports
HYPOTENSION908 reports
DYSPHAGIA900 reports
ARTHRALGIA897 reports
PRURITUS875 reports
SKIN DISCOLOURATION867 reports
THERAPY INTERRUPTED800 reports
NEUROTOXICITY787 reports
ASCITES776 reports
OEDEMA PERIPHERAL768 reports
PERIPHERAL SWELLING751 reports
URINARY TRACT INFECTION734 reports
RENAL FAILURE731 reports
HOSPITALISATION726 reports
MUSCLE SPASMS723 reports
BONE MARROW FAILURE716 reports
INTENTIONAL PRODUCT USE ISSUE714 reports
GAIT DISTURBANCE686 reports
DRUG INTOLERANCE685 reports
NO ADVERSE EVENT682 reports
GASTROINTESTINAL DISORDER675 reports
THROMBOSIS668 reports
HYPERSENSITIVITY663 reports
ABDOMINAL DISTENSION660 reports
ACUTE KIDNEY INJURY660 reports
PANCYTOPENIA658 reports
INTESTINAL OBSTRUCTION657 reports
BLOOD BILIRUBIN INCREASED653 reports
INSOMNIA653 reports
BLISTER647 reports
HAEMOGLOBIN DECREASED644 reports
EPISTAXIS637 reports
HEPATIC FUNCTION ABNORMAL635 reports
COLITIS634 reports
NEUTROPHIL COUNT DECREASED616 reports
PRODUCT USE IN UNAPPROVED INDICATION616 reports
CHILLS611 reports
CONFUSIONAL STATE598 reports
SKIN FISSURES597 reports

Key Safety Signals

  • High incidence of serious adverse reactions (82.2%)
  • Diverse range of reactions including neurological, gastrointestinal, and hematological issues
  • Significant number of reports involving disease progression and metastasis

Patient Demographics

Adverse event reports by sex: Female: 51,525, Male: 28,494, Unknown: 542. The most frequently reported age groups are age 65 (1,724 reports), age 66 (1,714 reports), age 70 (1,682 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 88,887 classified reports for CAPECITABINE:

  • Serious: 73,050 reports (82.2%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 15,837 reports (17.8%)
Serious 82.2%Non-Serious 17.8%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female51,525 (64.0%)
Male28,494 (35.4%)
Unknown542 (0.7%)

Reports by Age

Age 651,724 reports
Age 661,714 reports
Age 701,682 reports
Age 671,640 reports
Age 601,629 reports
Age 641,627 reports
Age 571,619 reports
Age 621,606 reports
Age 631,596 reports
Age 681,586 reports
Age 611,546 reports
Age 591,543 reports
Age 711,502 reports
Age 581,434 reports
Age 691,434 reports
Age 731,376 reports
Age 721,341 reports
Age 561,295 reports
Age 521,253 reports
Age 551,220 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Capecitabine can cause severe hematological and gastrointestinal side effects, and patients should be monitored closely for signs of toxicity. Drug interactions, particularly with other cytotoxic agents, should be avoided.

What You Should Know

If you are taking Capecitabine, here are important things to know. The most commonly reported side effects include diarrhoea, death, nausea, palmar-plantar erythrodysaesthesia syndrome, fatigue. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Monitor closely for signs of severe side effects such as severe diarrhea, nausea, and hematological issues. Follow healthcare provider’s guidance on managing side effects and adjusting dosages as necessary. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

Regulatory oversight is ongoing, with frequent updates to the drug’s labeling to include new safety information. Patients should report any adverse reactions immediately.

Frequently Asked Questions

How many adverse event reports has the FDA received for Capecitabine?

The FDA has received approximately 174,965 adverse event reports associated with Capecitabine. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Capecitabine?

The most frequently reported adverse events for Capecitabine include Diarrhoea, Death, Nausea, Palmar-Plantar Erythrodysaesthesia Syndrome, Fatigue. By volume, the top reported reactions are: Diarrhoea (13,395 reports), Death (8,723 reports), Nausea (8,248 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Capecitabine.

What percentage of Capecitabine adverse event reports are serious?

Out of 88,887 classified reports, 73,050 (82.2%) were classified as serious and 15,837 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Capecitabine (by sex)?

Adverse event reports for Capecitabine break down by patient sex as follows: Female: 51,525, Male: 28,494, Unknown: 542. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Capecitabine?

The most frequently reported age groups for Capecitabine adverse events are: age 65: 1,724 reports, age 66: 1,714 reports, age 70: 1,682 reports, age 67: 1,640 reports, age 60: 1,629 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Capecitabine?

The primary manufacturer associated with Capecitabine adverse event reports is H2-Pharma, Llc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Capecitabine?

Beyond the most common reactions, other reported adverse events for Capecitabine include: Vomiting, Disease Progression, Malignant Neoplasm Progression, Off Label Use, Asthenia. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Capecitabine?

You can report adverse events from Capecitabine to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Capecitabine's safety score and what does it mean?

Capecitabine has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Severe adverse reactions such as death, disease progression, and sepsis are frequently reported.

What are the key safety signals for Capecitabine?

Key safety signals identified in Capecitabine's adverse event data include: High incidence of serious adverse reactions (82.2%). Diverse range of reactions including neurological, gastrointestinal, and hematological issues. Significant number of reports involving disease progression and metastasis. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Capecitabine interact with other drugs?

Capecitabine can cause severe hematological and gastrointestinal side effects, and patients should be monitored closely for signs of toxicity. Drug interactions, particularly with other cytotoxic agents, should be avoided. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Capecitabine.

What should patients know before taking Capecitabine?

Monitor closely for signs of severe side effects such as severe diarrhea, nausea, and hematological issues. Follow healthcare provider’s guidance on managing side effects and adjusting dosages as necessary.

Are Capecitabine side effects well-documented?

Capecitabine has 174,965 adverse event reports on file with the FDA. Diarrhoea and nausea are the most common gastrointestinal side effects. The volume of reports for Capecitabine reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Capecitabine?

Regulatory oversight is ongoing, with frequent updates to the drug’s labeling to include new safety information. Patients should report any adverse reactions immediately. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to CAPECITABINE based on therapeutic use, drug class, or shared indications:

VincristineDocetaxelPaclitaxel
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.