IBRUTINIB

82/100 · Critical

Manufactured by Pharmacyclics LLC

High Serious Adverse Events with IBRUTINIB: Focus on Hematological and Cardiovascular Risks

129,122 FDA adverse event reports analyzed

Last updated: 2026-05-12

About IBRUTINIB

IBRUTINIB is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Pharmacyclics LLC. Based on analysis of 129,122 FDA adverse event reports, IBRUTINIB has a safety score of 82 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for IBRUTINIB include DEATH, OFF LABEL USE, FATIGUE, DIARRHOEA, ATRIAL FIBRILLATION. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for IBRUTINIB.

AI Safety Analysis

Ibrutinib has a safety concern score of 82 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 129,122 adverse event reports for this medication, which is primarily manufactured by Pharmacyclics Llc.

The most commonly reported adverse events include Death, Off Label Use, Fatigue. Of classified reports, 77.3% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. High incidence of serious adverse events, particularly hematological and cardiovascular issues.

Significant reports of infections and hematological abnormalities, including thrombocytopenia and neutropenia. Cardiovascular events such as atrial fibrillation and congestive heart failure are notable.

Patients taking Ibrutinib should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. IBRUTINIB can cause significant drug interactions, including those with warfarin and other anticoagulants, necessitating careful monitoring. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 82/100

Ibrutinib received a safety concern score of 82/100 (high concern). This is based on a 77.3% serious event ratio across 78,797 classified reports. The score accounts for 129,122 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

DEATH8,367 reports
OFF LABEL USE5,878 reports
FATIGUE4,668 reports
DIARRHOEA4,101 reports
ATRIAL FIBRILLATION3,797 reports
PNEUMONIA3,186 reports
CONTUSION2,778 reports
INCORRECT DOSE ADMINISTERED2,776 reports
FALL2,474 reports
ASTHENIA2,318 reports
NAUSEA2,272 reports
ARTHRALGIA2,179 reports
RASH2,118 reports
DISEASE PROGRESSION1,962 reports
HAEMORRHAGE1,960 reports
PYREXIA1,822 reports
MUSCLE SPASMS1,750 reports
COVID 191,712 reports
DIZZINESS1,708 reports
ANAEMIA1,663 reports
DYSPNOEA1,642 reports
PLATELET COUNT DECREASED1,619 reports
PAIN1,610 reports
HOSPITALISATION1,583 reports
PERIPHERAL SWELLING1,521 reports
HEADACHE1,509 reports
DRUG INEFFECTIVE1,493 reports
INFECTION1,446 reports
NEUTROPENIA1,436 reports
WHITE BLOOD CELL COUNT INCREASED1,431 reports
HYPERTENSION1,406 reports
THROMBOCYTOPENIA1,400 reports
URINARY TRACT INFECTION1,369 reports
WEIGHT DECREASED1,271 reports
PLEURAL EFFUSION1,243 reports
SURGERY1,231 reports
WHITE BLOOD CELL COUNT DECREASED1,198 reports
HAEMOGLOBIN DECREASED1,191 reports
PAIN IN EXTREMITY1,167 reports
COUGH1,163 reports
MALAISE1,158 reports
VOMITING1,126 reports
DECREASED APPETITE1,100 reports
MYALGIA1,091 reports
CONSTIPATION1,040 reports
EPISTAXIS1,031 reports
LYMPHADENOPATHY982 reports
PRODUCT USE IN UNAPPROVED INDICATION964 reports
SEPSIS955 reports
BACK PAIN954 reports
FEBRILE NEUTROPENIA952 reports
CATARACT945 reports
STOMATITIS884 reports
NASOPHARYNGITIS872 reports
CHRONIC LYMPHOCYTIC LEUKAEMIA867 reports
CARDIAC DISORDER864 reports
PRODUCT USE ISSUE783 reports
PRURITUS778 reports
ADVERSE DRUG REACTION738 reports
OEDEMA PERIPHERAL721 reports
DEHYDRATION719 reports
INSOMNIA714 reports
HYPOTENSION711 reports
INCREASED TENDENCY TO BRUISE704 reports
CEREBROVASCULAR ACCIDENT695 reports
BLOOD PRESSURE INCREASED656 reports
WEIGHT INCREASED653 reports
MYOCARDIAL INFARCTION651 reports
LOSS OF CONSCIOUSNESS632 reports
ONYCHOCLASIS630 reports
CARDIAC FAILURE CONGESTIVE612 reports
DYSPEPSIA611 reports
JOINT SWELLING609 reports
CARDIAC FAILURE598 reports
DRUG INTERACTION582 reports
NEUROPATHY PERIPHERAL578 reports
ACUTE KIDNEY INJURY576 reports
ABDOMINAL PAIN UPPER575 reports
CHEST PAIN572 reports
MEMORY IMPAIRMENT568 reports
FEELING ABNORMAL566 reports
ASPERGILLUS INFECTION542 reports
INFLUENZA537 reports
CYTOPENIA534 reports
SINUSITIS532 reports
ABDOMINAL DISCOMFORT530 reports
DEPRESSION526 reports
HOSPICE CARE514 reports
GAIT DISTURBANCE512 reports
PULMONARY OEDEMA512 reports
ABDOMINAL PAIN507 reports
HAEMATOMA502 reports
ANXIETY501 reports
DRY SKIN495 reports
PETECHIAE494 reports
BONE PAIN493 reports
PERICARDIAL EFFUSION492 reports
HAEMATURIA490 reports
CEREBRAL HAEMORRHAGE489 reports
PALPITATIONS485 reports

Key Safety Signals

  • Atrial fibrillation and other cardiac disorders are frequent.
  • Hematological issues like thrombocytopenia and neutropenia are common.
  • Infections, particularly pneumonia, are a significant concern.

Patient Demographics

Adverse event reports by sex: Male: 44,683, Female: 27,882, Unknown: 16. The most frequently reported age groups are age 74 (1,424 reports), age 75 (1,424 reports), age 70 (1,402 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 78,797 classified reports for IBRUTINIB:

  • Serious: 60,886 reports (77.3%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 17,911 reports (22.7%)
Serious 77.3%Non-Serious 22.7%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male44,683 (61.6%)
Female27,882 (38.4%)
Unknown16 (0.0%)

Reports by Age

Age 741,424 reports
Age 751,424 reports
Age 701,402 reports
Age 761,393 reports
Age 721,392 reports
Age 771,362 reports
Age 731,351 reports
Age 711,343 reports
Age 691,279 reports
Age 671,254 reports
Age 681,235 reports
Age 781,233 reports
Age 791,205 reports
Age 801,189 reports
Age 651,086 reports
Age 661,055 reports
Age 811,033 reports
Age 821,010 reports
Age 64993 reports
Age 83907 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

IBRUTINIB can cause significant drug interactions, including those with warfarin and other anticoagulants, necessitating careful monitoring.

What You Should Know

If you are taking Ibrutinib, here are important things to know. The most commonly reported side effects include death, off label use, fatigue, diarrhoea, atrial fibrillation. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Monitor for signs of infection, particularly in elderly patients, and report any symptoms promptly. Regularly check blood counts and monitor for hematological and cardiovascular adverse events. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

Regulatory oversight is ongoing, with regular updates on safety profiles and new warnings issued.

Frequently Asked Questions

How many adverse event reports has the FDA received for Ibrutinib?

The FDA has received approximately 129,122 adverse event reports associated with Ibrutinib. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Ibrutinib?

The most frequently reported adverse events for Ibrutinib include Death, Off Label Use, Fatigue, Diarrhoea, Atrial Fibrillation. By volume, the top reported reactions are: Death (8,367 reports), Off Label Use (5,878 reports), Fatigue (4,668 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Ibrutinib.

What percentage of Ibrutinib adverse event reports are serious?

Out of 78,797 classified reports, 60,886 (77.3%) were classified as serious and 17,911 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Ibrutinib (by sex)?

Adverse event reports for Ibrutinib break down by patient sex as follows: Male: 44,683, Female: 27,882, Unknown: 16. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Ibrutinib?

The most frequently reported age groups for Ibrutinib adverse events are: age 74: 1,424 reports, age 75: 1,424 reports, age 70: 1,402 reports, age 76: 1,393 reports, age 72: 1,392 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Ibrutinib?

The primary manufacturer associated with Ibrutinib adverse event reports is Pharmacyclics Llc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Ibrutinib?

Beyond the most common reactions, other reported adverse events for Ibrutinib include: Pneumonia, Contusion, Incorrect Dose Administered, Fall, Asthenia. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Ibrutinib?

You can report adverse events from Ibrutinib to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Ibrutinib's safety score and what does it mean?

Ibrutinib has a safety concern score of 82 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. High incidence of serious adverse events, particularly hematological and cardiovascular issues.

What are the key safety signals for Ibrutinib?

Key safety signals identified in Ibrutinib's adverse event data include: Atrial fibrillation and other cardiac disorders are frequent.. Hematological issues like thrombocytopenia and neutropenia are common.. Infections, particularly pneumonia, are a significant concern.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Ibrutinib interact with other drugs?

IBRUTINIB can cause significant drug interactions, including those with warfarin and other anticoagulants, necessitating careful monitoring. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Ibrutinib.

What should patients know before taking Ibrutinib?

Monitor for signs of infection, particularly in elderly patients, and report any symptoms promptly. Regularly check blood counts and monitor for hematological and cardiovascular adverse events.

Are Ibrutinib side effects well-documented?

Ibrutinib has 129,122 adverse event reports on file with the FDA. Significant reports of infections and hematological abnormalities, including thrombocytopenia and neutropenia. The volume of reports for Ibrutinib reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Ibrutinib?

Regulatory oversight is ongoing, with regular updates on safety profiles and new warnings issued. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to IBRUTINIB based on therapeutic use, drug class, or shared indications:

WarfarinAspirinCiprofloxacinRifampinIsoniazid
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.