LINAGLIPTIN

78/100 · Elevated

Manufactured by Boehringer Ingelheim Pharmaceuticals, Inc.

Linagliptin Adverse Events: High Serious Reaction Rate

46,358 FDA adverse event reports analyzed

Last updated: 2026-05-12

About LINAGLIPTIN

LINAGLIPTIN is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Boehringer Ingelheim Pharmaceuticals, Inc.. Based on analysis of 46,358 FDA adverse event reports, LINAGLIPTIN has a safety score of 78 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for LINAGLIPTIN include BLOOD GLUCOSE INCREASED, DIARRHOEA, NAUSEA, FATIGUE, DYSPNOEA. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for LINAGLIPTIN.

AI Safety Analysis

Linagliptin has a safety concern score of 78 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 46,358 adverse event reports for this medication, which is primarily manufactured by Boehringer Ingelheim Pharmaceuticals, Inc..

The most commonly reported adverse events include Blood Glucose Increased, Diarrhoea, Nausea. Of classified reports, 69.5% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. The most common reactions are gastrointestinal issues like nausea and diarrhea, indicating a potential for digestive side effects.

Serious reactions, such as acute kidney injury and myocardial infarction, are concerning and account for a significant portion of reports. A diverse range of reactions, including neurological and cardiovascular issues, suggests a broad safety profile.

Patients taking Linagliptin should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Linagliptin may interact with other drugs, including those affecting blood glucose levels, and warnings should be followed to avoid adverse effects. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 78/100

Linagliptin received a safety concern score of 78/100 (high concern). This is based on a 69.5% serious event ratio across 17,375 classified reports. The score accounts for 46,358 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

BLOOD GLUCOSE INCREASED1,326 reports
DIARRHOEA1,196 reports
NAUSEA1,138 reports
FATIGUE1,028 reports
DYSPNOEA998 reports
OFF LABEL USE921 reports
DIZZINESS919 reports
VOMITING875 reports
MALAISE789 reports
ACUTE KIDNEY INJURY772 reports
HEADACHE745 reports
ARTHRALGIA723 reports
PRURITUS720 reports
PYREXIA687 reports
DRUG INEFFECTIVE642 reports
PAIN641 reports
DEHYDRATION601 reports
ABDOMINAL PAIN UPPER600 reports
BACK PAIN599 reports
CHEST PAIN572 reports
ABDOMINAL DISCOMFORT558 reports
PERIPHERAL SWELLING558 reports
COVID 19553 reports
FALL548 reports
DEATH546 reports
INSOMNIA531 reports
MYOCARDIAL INFARCTION527 reports
ANXIETY523 reports
RASH512 reports
RENAL FAILURE498 reports
FEELING ABNORMAL496 reports
MUSCULAR WEAKNESS496 reports
ASTHENIA489 reports
PALPITATIONS488 reports
HYPERHIDROSIS479 reports
ALOPECIA473 reports
VISUAL IMPAIRMENT473 reports
CHRONIC KIDNEY DISEASE452 reports
MEMORY IMPAIRMENT451 reports
TACHYCARDIA450 reports
HEART RATE INCREASED445 reports
PNEUMONIA445 reports
WEIGHT DECREASED426 reports
HALLUCINATION422 reports
DRY SKIN420 reports
SUBARACHNOID HAEMORRHAGE412 reports
BLINDNESS408 reports
AMNESIA406 reports
ANGIOEDEMA404 reports
LIP SWELLING403 reports
INTENTIONAL PRODUCT MISUSE399 reports
TRANSIENT ISCHAEMIC ATTACK398 reports
DECREASED APPETITE393 reports
VENTRICULAR TACHYCARDIA391 reports
MIGRAINE385 reports
HYPOGLYCAEMIA384 reports
COGNITIVE DISORDER378 reports
TINNITUS372 reports
DISTURBANCE IN ATTENTION362 reports
EYE PRURITUS361 reports
CAROTID ARTERY OCCLUSION360 reports
PERICARDITIS360 reports
VASCULITIS360 reports
ATRIAL TACHYCARDIA358 reports
CARDIOSPASM356 reports
DIPLOPIA356 reports
MUSCLE TWITCHING356 reports
ANOSMIA354 reports
PRURITUS GENITAL354 reports
FACIAL PAIN353 reports
TENSION HEADACHE353 reports
PAIN OF SKIN352 reports
PALMOPLANTAR KERATODERMA349 reports
SLEEP TERROR349 reports
INTENTIONAL PRODUCT USE ISSUE346 reports
URINARY TRACT INFECTION336 reports
PANCREATITIS328 reports
HYPOTENSION321 reports
ABDOMINAL PAIN304 reports
COUGH296 reports
RENAL IMPAIRMENT295 reports
CONSTIPATION293 reports
PAIN IN EXTREMITY289 reports
GLYCOSYLATED HAEMOGLOBIN INCREASED286 reports
RASH PAPULAR262 reports
ANAEMIA249 reports
DRUG INTERACTION244 reports
IMMUNISATION244 reports
CARDIAC FAILURE242 reports
BLOOD PRESSURE INCREASED234 reports
PEMPHIGOID234 reports
HYPERGLYCAEMIA233 reports
HYPERTENSION232 reports
CONDITION AGGRAVATED230 reports
OEDEMA PERIPHERAL230 reports
CEREBROVASCULAR ACCIDENT215 reports
DERMATITIS BULLOUS213 reports
HYPERKALAEMIA213 reports
CONFUSIONAL STATE206 reports
DIABETES MELLITUS206 reports

Key Safety Signals

  • Acute kidney injury and myocardial infarction are key safety signals, indicating potential renal and cardiovascular risks.
  • Reports of falls and death highlight the need for careful patient monitoring, especially in elderly patients.
  • Drug ineffectiveness and hypoglycemia suggest potential issues with efficacy and blood glucose control.

Patient Demographics

Adverse event reports by sex: Female: 8,051, Male: 7,782, Unknown: 93. The most frequently reported age groups are age 70 (422 reports), age 71 (411 reports), age 75 (407 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 17,375 classified reports for LINAGLIPTIN:

  • Serious: 12,079 reports (69.5%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 5,296 reports (30.5%)
Serious 69.5%Non-Serious 30.5%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female8,051 (50.6%)
Male7,782 (48.9%)
Unknown93 (0.6%)

Reports by Age

Age 70422 reports
Age 71411 reports
Age 75407 reports
Age 73385 reports
Age 80362 reports
Age 72361 reports
Age 78349 reports
Age 69347 reports
Age 68342 reports
Age 74342 reports
Age 76337 reports
Age 77337 reports
Age 79329 reports
Age 65320 reports
Age 62309 reports
Age 67299 reports
Age 63295 reports
Age 81290 reports
Age 82290 reports
Age 66277 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Linagliptin may interact with other drugs, including those affecting blood glucose levels, and warnings should be followed to avoid adverse effects.

What You Should Know

If you are taking Linagliptin, here are important things to know. The most commonly reported side effects include blood glucose increased, diarrhoea, nausea, fatigue, dyspnoea. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Patients should be closely monitored for signs of serious reactions such as kidney injury or heart issues. Follow prescribed dosages and monitor blood glucose levels regularly to manage potential side effects. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA continues to monitor Linagliptin for safety, and updates will be provided as necessary. Healthcare providers should report any adverse events.

Frequently Asked Questions

How many adverse event reports has the FDA received for Linagliptin?

The FDA has received approximately 46,358 adverse event reports associated with Linagliptin. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Linagliptin?

The most frequently reported adverse events for Linagliptin include Blood Glucose Increased, Diarrhoea, Nausea, Fatigue, Dyspnoea. By volume, the top reported reactions are: Blood Glucose Increased (1,326 reports), Diarrhoea (1,196 reports), Nausea (1,138 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Linagliptin.

What percentage of Linagliptin adverse event reports are serious?

Out of 17,375 classified reports, 12,079 (69.5%) were classified as serious and 5,296 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Linagliptin (by sex)?

Adverse event reports for Linagliptin break down by patient sex as follows: Female: 8,051, Male: 7,782, Unknown: 93. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Linagliptin?

The most frequently reported age groups for Linagliptin adverse events are: age 70: 422 reports, age 71: 411 reports, age 75: 407 reports, age 73: 385 reports, age 80: 362 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Linagliptin?

The primary manufacturer associated with Linagliptin adverse event reports is Boehringer Ingelheim Pharmaceuticals, Inc.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Linagliptin?

Beyond the most common reactions, other reported adverse events for Linagliptin include: Off Label Use, Dizziness, Vomiting, Malaise, Acute Kidney Injury. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Linagliptin?

You can report adverse events from Linagliptin to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Linagliptin's safety score and what does it mean?

Linagliptin has a safety concern score of 78 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. The most common reactions are gastrointestinal issues like nausea and diarrhea, indicating a potential for digestive side effects.

What are the key safety signals for Linagliptin?

Key safety signals identified in Linagliptin's adverse event data include: Acute kidney injury and myocardial infarction are key safety signals, indicating potential renal and cardiovascular risks.. Reports of falls and death highlight the need for careful patient monitoring, especially in elderly patients.. Drug ineffectiveness and hypoglycemia suggest potential issues with efficacy and blood glucose control.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Linagliptin interact with other drugs?

Linagliptin may interact with other drugs, including those affecting blood glucose levels, and warnings should be followed to avoid adverse effects. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Linagliptin.

What should patients know before taking Linagliptin?

Patients should be closely monitored for signs of serious reactions such as kidney injury or heart issues. Follow prescribed dosages and monitor blood glucose levels regularly to manage potential side effects.

Are Linagliptin side effects well-documented?

Linagliptin has 46,358 adverse event reports on file with the FDA. Serious reactions, such as acute kidney injury and myocardial infarction, are concerning and account for a significant portion of reports. The volume of reports for Linagliptin reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Linagliptin?

The FDA continues to monitor Linagliptin for safety, and updates will be provided as necessary. Healthcare providers should report any adverse events. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to LINAGLIPTIN based on therapeutic use, drug class, or shared indications:

MetforminSulfonylureasInsulin
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.