LINEZOLID

85/100 · Critical

Manufactured by Hp Halden Pharma AS

Linezolid Adverse Events: High Seriousness and Diverse Reactions

47,534 FDA adverse event reports analyzed

Last updated: 2026-05-12

About LINEZOLID

LINEZOLID is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Hp Halden Pharma AS. Based on analysis of 47,534 FDA adverse event reports, LINEZOLID has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for LINEZOLID include OFF LABEL USE, THROMBOCYTOPENIA, DRUG INEFFECTIVE, ANAEMIA, DRUG INTERACTION. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for LINEZOLID.

AI Safety Analysis

Linezolid has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 47,534 adverse event reports for this medication, which is primarily manufactured by Hp Halden Pharma As.

The most commonly reported adverse events include Off Label Use, Thrombocytopenia, Drug Ineffective. Of classified reports, 90.6% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Linezolid reports show a high percentage of serious adverse events, with over 90% of reported outcomes being serious.

The drug is associated with a wide range of reactions, including neurological, hematological, and gastrointestinal issues. Death and severe infections are among the most reported serious adverse events.

Patients taking Linezolid should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Linezolid can interact with other drugs, leading to potential toxicity. Warnings include interactions with drugs that affect QT interval and those that can cause bone marrow suppression. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Linezolid received a safety concern score of 85/100 (high concern). This is based on a 90.6% serious event ratio across 27,999 classified reports. The score accounts for 47,534 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

OFF LABEL USE2,426 reports
THROMBOCYTOPENIA2,032 reports
DRUG INEFFECTIVE1,993 reports
ANAEMIA1,601 reports
DRUG INTERACTION1,383 reports
NAUSEA1,301 reports
VOMITING1,063 reports
DIARRHOEA1,003 reports
PLATELET COUNT DECREASED999 reports
PYREXIA981 reports
LACTIC ACIDOSIS938 reports
NEUROPATHY PERIPHERAL901 reports
SEROTONIN SYNDROME874 reports
ACUTE KIDNEY INJURY867 reports
PANCYTOPENIA853 reports
DEATH759 reports
DRUG RESISTANCE729 reports
CONDITION AGGRAVATED728 reports
DYSPNOEA722 reports
PNEUMONIA701 reports
ELECTROCARDIOGRAM QT PROLONGED697 reports
SEPSIS681 reports
PRODUCT USE IN UNAPPROVED INDICATION673 reports
SEPTIC SHOCK611 reports
RESPIRATORY FAILURE602 reports
ASTHENIA545 reports
RASH541 reports
RENAL FAILURE503 reports
HYPOTENSION498 reports
TOXICITY TO VARIOUS AGENTS469 reports
MULTIPLE ORGAN DYSFUNCTION SYNDROME468 reports
DECREASED APPETITE450 reports
RENAL IMPAIRMENT442 reports
HAEMOGLOBIN DECREASED433 reports
NEUTROPENIA429 reports
CONFUSIONAL STATE428 reports
DIZZINESS386 reports
TREATMENT FAILURE378 reports
HEADACHE371 reports
FATIGUE358 reports
DRUG REACTION WITH EOSINOPHILIA AND SYSTEMIC SYMPTOMS353 reports
STAPHYLOCOCCAL INFECTION349 reports
MALAISE345 reports
ABDOMINAL PAIN335 reports
WEIGHT DECREASED333 reports
MYELOSUPPRESSION330 reports
HYPONATRAEMIA324 reports
PATHOGEN RESISTANCE323 reports
PRODUCT USE ISSUE317 reports
INFECTION312 reports
HEPATOTOXICITY310 reports
DRUG INEFFECTIVE FOR UNAPPROVED INDICATION296 reports
LEUKOPENIA294 reports
BONE MARROW FAILURE292 reports
HYPOKALAEMIA288 reports
BLOOD CREATININE INCREASED271 reports
WHITE BLOOD CELL COUNT DECREASED271 reports
GENERAL PHYSICAL HEALTH DETERIORATION263 reports
HYPERTENSION263 reports
DRUG HYPERSENSITIVITY262 reports
PRURITUS260 reports
DRUG INTOLERANCE258 reports
DRUG INDUCED LIVER INJURY258 reports
ALANINE AMINOTRANSFERASE INCREASED257 reports
GASTROINTESTINAL DISORDER256 reports
PAIN250 reports
ASPARTATE AMINOTRANSFERASE INCREASED238 reports
COUGH237 reports
ARTHRALGIA236 reports
ERYTHEMA232 reports
HYPOGLYCAEMIA232 reports
HYPOAESTHESIA230 reports
TACHYCARDIA228 reports
PARAESTHESIA226 reports
EOSINOPHILIA222 reports
OPTIC NEUROPATHY222 reports
TREMOR222 reports
GASTROINTESTINAL HAEMORRHAGE218 reports
INTENTIONAL PRODUCT USE ISSUE216 reports
METABOLIC ACIDOSIS212 reports
CARDIAC ARREST208 reports
ANXIETY207 reports
FEBRILE NEUTROPENIA206 reports
CARDIAC FAILURE205 reports
DISEASE PROGRESSION203 reports
ENTEROCOCCAL INFECTION203 reports
HALLUCINATION202 reports
RASH MACULO PAPULAR202 reports
HEPATIC FAILURE199 reports
HYPERSENSITIVITY197 reports
PLEURAL EFFUSION192 reports
TUBERCULOSIS190 reports
URINARY TRACT INFECTION187 reports
VISION BLURRED186 reports
VISUAL IMPAIRMENT186 reports
RENAL FAILURE ACUTE183 reports
DEHYDRATION182 reports
SEIZURE182 reports
CONSTIPATION178 reports
DEPRESSION178 reports

Key Safety Signals

  • Serious adverse events (25,361 out of 27,999) make up over 90% of the total reported outcomes.
  • Neurological issues such as peripheral neuropathy and serotonin syndrome are key safety signals.
  • Hematological issues like pancytopenia and thrombocytopenia are also significant safety signals.

Patient Demographics

Adverse event reports by sex: Male: 13,828, Female: 10,735, Unknown: 180. The most frequently reported age groups are age 65 (496 reports), age 70 (495 reports), age 67 (455 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 27,999 classified reports for LINEZOLID:

  • Serious: 25,361 reports (90.6%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 2,638 reports (9.4%)
Serious 90.6%Non-Serious 9.4%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male13,828 (55.9%)
Female10,735 (43.4%)
Unknown180 (0.7%)

Reports by Age

Age 65496 reports
Age 70495 reports
Age 67455 reports
Age 60441 reports
Age 66437 reports
Age 69421 reports
Age 57409 reports
Age 68405 reports
Age 64402 reports
Age 58399 reports
Age 75393 reports
Age 63390 reports
Age 76389 reports
Age 71388 reports
Age 72382 reports
Age 56380 reports
Age 73379 reports
Age 61358 reports
Age 59335 reports
Age 74333 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Linezolid can interact with other drugs, leading to potential toxicity. Warnings include interactions with drugs that affect QT interval and those that can cause bone marrow suppression.

What You Should Know

If you are taking Linezolid, here are important things to know. The most commonly reported side effects include off label use, thrombocytopenia, drug ineffective, anaemia, drug interaction. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Patients should report any new or worsening symptoms to their healthcare provider immediately. Follow all prescribed dosages and do not alter the treatment without medical advice. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA continues to monitor Linezolid for safety, particularly for serious adverse events and drug interactions. Healthcare providers should be vigilant and report any adverse events.

Frequently Asked Questions

How many adverse event reports has the FDA received for Linezolid?

The FDA has received approximately 47,534 adverse event reports associated with Linezolid. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Linezolid?

The most frequently reported adverse events for Linezolid include Off Label Use, Thrombocytopenia, Drug Ineffective, Anaemia, Drug Interaction. By volume, the top reported reactions are: Off Label Use (2,426 reports), Thrombocytopenia (2,032 reports), Drug Ineffective (1,993 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Linezolid.

What percentage of Linezolid adverse event reports are serious?

Out of 27,999 classified reports, 25,361 (90.6%) were classified as serious and 2,638 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Linezolid (by sex)?

Adverse event reports for Linezolid break down by patient sex as follows: Male: 13,828, Female: 10,735, Unknown: 180. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Linezolid?

The most frequently reported age groups for Linezolid adverse events are: age 65: 496 reports, age 70: 495 reports, age 67: 455 reports, age 60: 441 reports, age 66: 437 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Linezolid?

The primary manufacturer associated with Linezolid adverse event reports is Hp Halden Pharma As. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Linezolid?

Beyond the most common reactions, other reported adverse events for Linezolid include: Nausea, Vomiting, Diarrhoea, Platelet Count Decreased, Pyrexia. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Linezolid?

You can report adverse events from Linezolid to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Linezolid's safety score and what does it mean?

Linezolid has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Linezolid reports show a high percentage of serious adverse events, with over 90% of reported outcomes being serious.

What are the key safety signals for Linezolid?

Key safety signals identified in Linezolid's adverse event data include: Serious adverse events (25,361 out of 27,999) make up over 90% of the total reported outcomes.. Neurological issues such as peripheral neuropathy and serotonin syndrome are key safety signals.. Hematological issues like pancytopenia and thrombocytopenia are also significant safety signals.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Linezolid interact with other drugs?

Linezolid can interact with other drugs, leading to potential toxicity. Warnings include interactions with drugs that affect QT interval and those that can cause bone marrow suppression. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Linezolid.

What should patients know before taking Linezolid?

Patients should report any new or worsening symptoms to their healthcare provider immediately. Follow all prescribed dosages and do not alter the treatment without medical advice.

Are Linezolid side effects well-documented?

Linezolid has 47,534 adverse event reports on file with the FDA. The drug is associated with a wide range of reactions, including neurological, hematological, and gastrointestinal issues. The volume of reports for Linezolid reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Linezolid?

The FDA continues to monitor Linezolid for safety, particularly for serious adverse events and drug interactions. Healthcare providers should be vigilant and report any adverse events. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to LINEZOLID based on therapeutic use, drug class, or shared indications:

DoxycyclineCiprofloxacinAmphotericin BVancomycinFluconazole
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.