LOPERAMIDE HYDROCHLORIDE

72/100 · Elevated

Manufactured by Kenvue Brands LLC

High Incidence of Gastrointestinal and General Symptoms with Loperamide Hydrochloride

100,013 FDA adverse event reports analyzed

Last updated: 2026-05-12

About LOPERAMIDE HYDROCHLORIDE

LOPERAMIDE HYDROCHLORIDE is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Kenvue Brands LLC. Based on analysis of 100,013 FDA adverse event reports, LOPERAMIDE HYDROCHLORIDE has a safety score of 72 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for LOPERAMIDE HYDROCHLORIDE include DIARRHOEA, NAUSEA, DRUG INEFFECTIVE, FATIGUE, OFF LABEL USE. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for LOPERAMIDE HYDROCHLORIDE.

AI Safety Analysis

Loperamide Hydrochloride has a safety concern score of 72 out of 100, placing it in the elevated concern category based on analysis of FDA adverse event data. The FDA has received approximately 100,013 adverse event reports for this medication, which is primarily manufactured by Kenvue Brands Llc.

The most commonly reported adverse events include Diarrhoea, Nausea, Drug Ineffective. Of classified reports, 61.6% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Gastrointestinal symptoms such as diarrhea, nausea, and abdominal pain are frequently reported.

General symptoms like fatigue, dizziness, and headache are also common. Serious adverse events, including pneumonia and death, are reported but less frequently.

Patients taking Loperamide Hydrochloride should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Loperamide Hydrochloride can cause gastrointestinal issues and should be used with caution, especially in combination with other drugs that affect the gastrointestinal tract. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 72/100

Loperamide Hydrochloride received a safety concern score of 72/100 (elevated concern). This is based on a 61.6% serious event ratio across 42,604 classified reports. The score accounts for 100,013 total adverse event reports and 100 distinct reaction types. This elevated score indicates a notable proportion of serious adverse events and warrants careful monitoring.

Top Adverse Reactions

DIARRHOEA8,465 reports
NAUSEA4,090 reports
DRUG INEFFECTIVE3,914 reports
FATIGUE3,690 reports
OFF LABEL USE3,095 reports
VOMITING2,673 reports
CONSTIPATION2,352 reports
WEIGHT DECREASED2,018 reports
HEADACHE1,891 reports
DYSPNOEA1,881 reports
ABDOMINAL PAIN1,757 reports
ASTHENIA1,743 reports
DECREASED APPETITE1,712 reports
DIZZINESS1,615 reports
PAIN1,596 reports
PNEUMONIA1,546 reports
DEHYDRATION1,534 reports
PYREXIA1,503 reports
MALAISE1,389 reports
INCORRECT DOSE ADMINISTERED1,329 reports
DEATH1,283 reports
COUGH1,241 reports
ARTHRALGIA1,223 reports
RASH1,155 reports
ABDOMINAL PAIN UPPER1,132 reports
INTENTIONAL PRODUCT USE ISSUE1,102 reports
ANAEMIA1,098 reports
FALL1,038 reports
PAIN IN EXTREMITY1,009 reports
BACK PAIN895 reports
ABDOMINAL DISCOMFORT881 reports
SOMNOLENCE837 reports
CONDITION AGGRAVATED831 reports
URINARY TRACT INFECTION822 reports
PRURITUS812 reports
HYPOTENSION811 reports
GASTROOESOPHAGEAL REFLUX DISEASE773 reports
INSOMNIA756 reports
ABDOMINAL DISTENSION740 reports
MUSCLE SPASMS713 reports
HYPERTENSION700 reports
DYSPEPSIA698 reports
BLOOD PRESSURE INCREASED686 reports
PERIPHERAL SWELLING686 reports
ACUTE KIDNEY INJURY678 reports
OEDEMA PERIPHERAL678 reports
OVERDOSE667 reports
FLATULENCE666 reports
INAPPROPRIATE SCHEDULE OF PRODUCT ADMINISTRATION659 reports
NASOPHARYNGITIS651 reports
PRODUCT DOSE OMISSION ISSUE646 reports
WEIGHT INCREASED639 reports
EXPIRED PRODUCT ADMINISTERED620 reports
PRODUCT USE IN UNAPPROVED INDICATION601 reports
ANXIETY600 reports
CHEST PAIN597 reports
FEELING ABNORMAL579 reports
PRODUCT USE ISSUE575 reports
PLATELET COUNT DECREASED552 reports
SEPSIS546 reports
HAEMOGLOBIN DECREASED540 reports
NEUTROPENIA540 reports
ALOPECIA530 reports
WHITE BLOOD CELL COUNT DECREASED527 reports
INCORRECT PRODUCT ADMINISTRATION DURATION525 reports
HAEMATOCHEZIA516 reports
ERYTHEMA507 reports
CROHN^S DISEASE499 reports
FREQUENT BOWEL MOVEMENTS498 reports
HYPOKALAEMIA495 reports
COLITIS489 reports
COVID 19488 reports
GAIT DISTURBANCE485 reports
DEPRESSION483 reports
CONFUSIONAL STATE475 reports
CHILLS471 reports
INTENTIONAL PRODUCT MISUSE464 reports
DYSPHAGIA460 reports
STOMATITIS456 reports
DISEASE PROGRESSION454 reports
INFECTION454 reports
GASTROINTESTINAL DISORDER451 reports
RENAL FAILURE451 reports
COMA447 reports
MYALGIA435 reports
NEUROPATHY PERIPHERAL434 reports
THROMBOCYTOPENIA433 reports
MALIGNANT NEOPLASM PROGRESSION430 reports
FEBRILE NEUTROPENIA427 reports
SYNCOPE425 reports
DRY SKIN419 reports
HYPOAESTHESIA419 reports
BLOOD CREATININE INCREASED418 reports
PNEUMONIA ASPIRATION410 reports
ATRIAL FIBRILLATION408 reports
OROPHARYNGEAL PAIN403 reports
DRUG INTERACTION398 reports
HYPERSENSITIVITY398 reports
INTESTINAL OBSTRUCTION391 reports
TREMOR391 reports

Key Safety Signals

  • Diarrhea and nausea are the most common reactions.
  • Reports of serious events like pneumonia and death indicate potential severe risks.
  • Off-label use and incorrect dose administration are significant safety signals.

Patient Demographics

Adverse event reports by sex: Female: 24,240, Male: 14,741, Unknown: 25. The most frequently reported age groups are age 64 (869 reports), age 72 (763 reports), age 69 (761 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 42,604 classified reports for LOPERAMIDE HYDROCHLORIDE:

  • Serious: 26,264 reports (61.6%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 16,340 reports (38.4%)
Serious 61.6%Non-Serious 38.4%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female24,240 (62.1%)
Male14,741 (37.8%)
Unknown25 (0.1%)

Reports by Age

Age 64869 reports
Age 72763 reports
Age 69761 reports
Age 75759 reports
Age 71756 reports
Age 73746 reports
Age 67730 reports
Age 74728 reports
Age 68712 reports
Age 70705 reports
Age 65704 reports
Age 66669 reports
Age 62650 reports
Age 76643 reports
Age 77613 reports
Age 63589 reports
Age 78574 reports
Age 60562 reports
Age 59554 reports
Age 52539 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Loperamide Hydrochloride can cause gastrointestinal issues and should be used with caution, especially in combination with other drugs that affect the gastrointestinal tract.

What You Should Know

If you are taking Loperamide Hydrochloride, here are important things to know. The most commonly reported side effects include diarrhoea, nausea, drug ineffective, fatigue, off label use. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Follow prescribed dosages and do not exceed recommended limits. Report any serious adverse events to healthcare providers immediately. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA closely monitors Loperamide Hydrochloride due to its potential for serious adverse events, particularly in higher doses or off-label use.

Frequently Asked Questions

How many adverse event reports has the FDA received for Loperamide Hydrochloride?

The FDA has received approximately 100,013 adverse event reports associated with Loperamide Hydrochloride. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Loperamide Hydrochloride?

The most frequently reported adverse events for Loperamide Hydrochloride include Diarrhoea, Nausea, Drug Ineffective, Fatigue, Off Label Use. By volume, the top reported reactions are: Diarrhoea (8,465 reports), Nausea (4,090 reports), Drug Ineffective (3,914 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Loperamide Hydrochloride.

What percentage of Loperamide Hydrochloride adverse event reports are serious?

Out of 42,604 classified reports, 26,264 (61.6%) were classified as serious and 16,340 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Loperamide Hydrochloride (by sex)?

Adverse event reports for Loperamide Hydrochloride break down by patient sex as follows: Female: 24,240, Male: 14,741, Unknown: 25. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Loperamide Hydrochloride?

The most frequently reported age groups for Loperamide Hydrochloride adverse events are: age 64: 869 reports, age 72: 763 reports, age 69: 761 reports, age 75: 759 reports, age 71: 756 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Loperamide Hydrochloride?

The primary manufacturer associated with Loperamide Hydrochloride adverse event reports is Kenvue Brands Llc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Loperamide Hydrochloride?

Beyond the most common reactions, other reported adverse events for Loperamide Hydrochloride include: Vomiting, Constipation, Weight Decreased, Headache, Dyspnoea. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Loperamide Hydrochloride?

You can report adverse events from Loperamide Hydrochloride to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Loperamide Hydrochloride's safety score and what does it mean?

Loperamide Hydrochloride has a safety concern score of 72 out of 100 (elevated concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Gastrointestinal symptoms such as diarrhea, nausea, and abdominal pain are frequently reported.

What are the key safety signals for Loperamide Hydrochloride?

Key safety signals identified in Loperamide Hydrochloride's adverse event data include: Diarrhea and nausea are the most common reactions.. Reports of serious events like pneumonia and death indicate potential severe risks.. Off-label use and incorrect dose administration are significant safety signals.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Loperamide Hydrochloride interact with other drugs?

Loperamide Hydrochloride can cause gastrointestinal issues and should be used with caution, especially in combination with other drugs that affect the gastrointestinal tract. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Loperamide Hydrochloride.

What should patients know before taking Loperamide Hydrochloride?

Follow prescribed dosages and do not exceed recommended limits. Report any serious adverse events to healthcare providers immediately.

Are Loperamide Hydrochloride side effects well-documented?

Loperamide Hydrochloride has 100,013 adverse event reports on file with the FDA. General symptoms like fatigue, dizziness, and headache are also common. The volume of reports for Loperamide Hydrochloride reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Loperamide Hydrochloride?

The FDA closely monitors Loperamide Hydrochloride due to its potential for serious adverse events, particularly in higher doses or off-label use. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to LOPERAMIDE HYDROCHLORIDE based on therapeutic use, drug class, or shared indications:

CodeineTramadolOxycodone
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.