MYCOPHENOLATE MOFETIL

85/100 · Critical

Manufactured by Genentech, Inc.

Mycophenolate Mofetil Adverse Events: High Seriousness and Diverse Reactions

256,184 FDA adverse event reports analyzed

Last updated: 2026-05-12

About MYCOPHENOLATE MOFETIL

MYCOPHENOLATE MOFETIL is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Genentech, Inc.. Based on analysis of 256,184 FDA adverse event reports, MYCOPHENOLATE MOFETIL has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for MYCOPHENOLATE MOFETIL include OFF LABEL USE, DRUG INEFFECTIVE, PRODUCT USE IN UNAPPROVED INDICATION, DIARRHOEA, PYREXIA. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for MYCOPHENOLATE MOFETIL.

AI Safety Analysis

Mycophenolate Mofetil has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 256,184 adverse event reports for this medication, which is primarily manufactured by Genentech, Inc..

The most commonly reported adverse events include Off Label Use, Drug Ineffective, Product Use In Unapproved Indication. Of classified reports, 91.5% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. High percentage of serious adverse events (91.5%) indicates significant safety concerns.

Diverse range of reactions, including infections, renal impairment, and graft rejection, highlight the drug's broad potential risks. Report volume is substantial, with over 256,000 reports, providing a comprehensive dataset for analysis.

Patients taking Mycophenolate Mofetil should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Mycophenolate Mofetil can interact with other immunosuppressants and may increase the risk of infections and other adverse events. Warnings include monitoring for drug interactions and infections. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Mycophenolate Mofetil received a safety concern score of 85/100 (high concern). This is based on a 91.5% serious event ratio across 128,019 classified reports. The score accounts for 256,184 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

OFF LABEL USE17,971 reports
DRUG INEFFECTIVE10,593 reports
PRODUCT USE IN UNAPPROVED INDICATION7,053 reports
DIARRHOEA6,605 reports
PYREXIA5,434 reports
PNEUMONIA5,027 reports
CYTOMEGALOVIRUS INFECTION4,729 reports
NAUSEA4,256 reports
FATIGUE4,238 reports
CONDITION AGGRAVATED4,176 reports
TRANSPLANT REJECTION4,029 reports
DYSPNOEA3,886 reports
VOMITING3,865 reports
HEADACHE3,704 reports
ACUTE KIDNEY INJURY3,631 reports
INFECTION3,551 reports
COVID 193,388 reports
SEPSIS3,254 reports
DEATH3,237 reports
DRUG INTERACTION3,219 reports
HYPERTENSION3,138 reports
RASH2,831 reports
INTENTIONAL PRODUCT USE ISSUE2,791 reports
ARTHRALGIA2,746 reports
MALAISE2,701 reports
ASTHENIA2,691 reports
PAIN2,680 reports
TREATMENT FAILURE2,679 reports
RENAL IMPAIRMENT2,611 reports
ANAEMIA2,605 reports
WEIGHT DECREASED2,575 reports
DRUG INTOLERANCE2,484 reports
NEUTROPENIA2,423 reports
RESPIRATORY FAILURE2,311 reports
LEUKOPENIA2,273 reports
WEIGHT INCREASED2,267 reports
URINARY TRACT INFECTION2,257 reports
COUGH2,227 reports
DECREASED APPETITE2,196 reports
BLOOD CREATININE INCREASED2,184 reports
SEPTIC SHOCK2,182 reports
ABDOMINAL PAIN2,177 reports
SYSTEMIC LUPUS ERYTHEMATOSUS2,112 reports
DRUG INEFFECTIVE FOR UNAPPROVED INDICATION2,107 reports
DIZZINESS2,103 reports
ALOPECIA2,102 reports
POST TRANSPLANT LYMPHOPROLIFERATIVE DISORDER2,090 reports
TOXICITY TO VARIOUS AGENTS2,081 reports
PRURITUS2,053 reports
GASTROINTESTINAL DISORDER1,962 reports
RHEUMATOID ARTHRITIS1,960 reports
RENAL FAILURE1,942 reports
GENERAL PHYSICAL HEALTH DETERIORATION1,933 reports
THROMBOCYTOPENIA1,929 reports
SINUSITIS1,920 reports
MULTIPLE ORGAN DYSFUNCTION SYNDROME1,917 reports
JOINT SWELLING1,880 reports
KIDNEY TRANSPLANT REJECTION1,843 reports
ABDOMINAL DISCOMFORT1,795 reports
PANCYTOPENIA1,771 reports
THERAPY NON RESPONDER1,751 reports
HYPOAESTHESIA1,733 reports
INFUSION RELATED REACTION1,691 reports
CONFUSIONAL STATE1,689 reports
ABDOMINAL PAIN UPPER1,646 reports
DRUG HYPERSENSITIVITY1,638 reports
PRODUCT USE ISSUE1,637 reports
CHEST PAIN1,631 reports
NASOPHARYNGITIS1,616 reports
PSORIATIC ARTHROPATHY1,615 reports
HYPERSENSITIVITY1,605 reports
THROMBOTIC MICROANGIOPATHY1,603 reports
HEPATIC ENZYME INCREASED1,560 reports
INSOMNIA1,546 reports
OEDEMA1,534 reports
EPSTEIN BARR VIRUS INFECTION1,523 reports
SWELLING1,506 reports
PERIPHERAL SWELLING1,498 reports
OEDEMA PERIPHERAL1,485 reports
MATERNAL EXPOSURE DURING PREGNANCY1,477 reports
DISEASE PROGRESSION1,474 reports
STOMATITIS1,470 reports
PAIN IN EXTREMITY1,466 reports
SCIATICA1,450 reports
MOBILITY DECREASED1,439 reports
CYTOMEGALOVIRUS VIRAEMIA1,421 reports
SYNOVITIS1,402 reports
URTICARIA1,398 reports
BK VIRUS INFECTION1,392 reports
TYPE 2 DIABETES MELLITUS1,389 reports
GRAFT VERSUS HOST DISEASE1,388 reports
ACUTE GRAFT VERSUS HOST DISEASE1,386 reports
IMPAIRED HEALING1,386 reports
HYPOTENSION1,362 reports
POLYOMAVIRUS ASSOCIATED NEPHROPATHY1,356 reports
LUNG DISORDER1,354 reports
ANXIETY1,343 reports
FIBROMYALGIA1,332 reports
MUSCULOSKELETAL STIFFNESS1,330 reports
PEMPHIGUS1,287 reports

Key Safety Signals

  • High incidence of infections (Pneumonia, Cytomegalovirus Infection, Sepsis, etc.)
  • Renal impairment and failure are frequently reported, indicating potential nephrotoxicity.
  • Graft rejection and transplant complications are significant concerns, especially in transplant patients.

Patient Demographics

Adverse event reports by sex: Male: 55,598, Female: 54,295, Unknown: 644. The most frequently reported age groups are age 43 (2,507 reports), age 44 (2,224 reports), age 60 (2,199 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 128,019 classified reports for MYCOPHENOLATE MOFETIL:

  • Serious: 117,114 reports (91.5%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 10,905 reports (8.5%)
Serious 91.5%Non-Serious 8.5%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male55,598 (50.3%)
Female54,295 (49.1%)
Unknown644 (0.6%)

Reports by Age

Age 432,507 reports
Age 442,224 reports
Age 602,199 reports
Age 572,132 reports
Age 552,073 reports
Age 642,068 reports
Age 581,991 reports
Age 561,988 reports
Age 591,984 reports
Age 631,941 reports
Age 501,920 reports
Age 621,918 reports
Age 611,915 reports
Age 531,868 reports
Age 451,858 reports
Age 521,828 reports
Age 541,803 reports
Age 651,789 reports
Age 661,758 reports
Age 511,647 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Mycophenolate Mofetil can interact with other immunosuppressants and may increase the risk of infections and other adverse events. Warnings include monitoring for drug interactions and infections.

What You Should Know

If you are taking Mycophenolate Mofetil, here are important things to know. The most commonly reported side effects include off label use, drug ineffective, product use in unapproved indication, diarrhoea, pyrexia. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Patients should report any new or worsening symptoms to their healthcare provider immediately. Regular monitoring for signs of infection, renal function, and graft rejection is crucial. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA continues to monitor Mycophenolate Mofetil for safety, and updates are regularly issued based on new data. Healthcare providers should stay informed about the latest safety information.

Frequently Asked Questions

How many adverse event reports has the FDA received for Mycophenolate Mofetil?

The FDA has received approximately 256,184 adverse event reports associated with Mycophenolate Mofetil. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Mycophenolate Mofetil?

The most frequently reported adverse events for Mycophenolate Mofetil include Off Label Use, Drug Ineffective, Product Use In Unapproved Indication, Diarrhoea, Pyrexia. By volume, the top reported reactions are: Off Label Use (17,971 reports), Drug Ineffective (10,593 reports), Product Use In Unapproved Indication (7,053 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Mycophenolate Mofetil.

What percentage of Mycophenolate Mofetil adverse event reports are serious?

Out of 128,019 classified reports, 117,114 (91.5%) were classified as serious and 10,905 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Mycophenolate Mofetil (by sex)?

Adverse event reports for Mycophenolate Mofetil break down by patient sex as follows: Male: 55,598, Female: 54,295, Unknown: 644. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Mycophenolate Mofetil?

The most frequently reported age groups for Mycophenolate Mofetil adverse events are: age 43: 2,507 reports, age 44: 2,224 reports, age 60: 2,199 reports, age 57: 2,132 reports, age 55: 2,073 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Mycophenolate Mofetil?

The primary manufacturer associated with Mycophenolate Mofetil adverse event reports is Genentech, Inc.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Mycophenolate Mofetil?

Beyond the most common reactions, other reported adverse events for Mycophenolate Mofetil include: Pneumonia, Cytomegalovirus Infection, Nausea, Fatigue, Condition Aggravated. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Mycophenolate Mofetil?

You can report adverse events from Mycophenolate Mofetil to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Mycophenolate Mofetil's safety score and what does it mean?

Mycophenolate Mofetil has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. High percentage of serious adverse events (91.5%) indicates significant safety concerns.

What are the key safety signals for Mycophenolate Mofetil?

Key safety signals identified in Mycophenolate Mofetil's adverse event data include: High incidence of infections (Pneumonia, Cytomegalovirus Infection, Sepsis, etc.). Renal impairment and failure are frequently reported, indicating potential nephrotoxicity.. Graft rejection and transplant complications are significant concerns, especially in transplant patients.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Mycophenolate Mofetil interact with other drugs?

Mycophenolate Mofetil can interact with other immunosuppressants and may increase the risk of infections and other adverse events. Warnings include monitoring for drug interactions and infections. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Mycophenolate Mofetil.

What should patients know before taking Mycophenolate Mofetil?

Patients should report any new or worsening symptoms to their healthcare provider immediately. Regular monitoring for signs of infection, renal function, and graft rejection is crucial.

Are Mycophenolate Mofetil side effects well-documented?

Mycophenolate Mofetil has 256,184 adverse event reports on file with the FDA. Diverse range of reactions, including infections, renal impairment, and graft rejection, highlight the drug's broad potential risks. The volume of reports for Mycophenolate Mofetil reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Mycophenolate Mofetil?

The FDA continues to monitor Mycophenolate Mofetil for safety, and updates are regularly issued based on new data. Healthcare providers should stay informed about the latest safety information. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to MYCOPHENOLATE MOFETIL based on therapeutic use, drug class, or shared indications:

CyclosporineTacrolimusPrednisone
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.