TENOFOVIR DISOPROXIL FUMARATE

85/100 · Critical

Manufactured by Gilead Sciences, Inc.

High Safety Concerns with Tenofovir Disoproxil Fumarate, Particularly for Bone and Renal Health

123,510 FDA adverse event reports analyzed

Last updated: 2026-05-12

About TENOFOVIR DISOPROXIL FUMARATE

TENOFOVIR DISOPROXIL FUMARATE is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Gilead Sciences, Inc.. Based on analysis of 123,510 FDA adverse event reports, TENOFOVIR DISOPROXIL FUMARATE has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for TENOFOVIR DISOPROXIL FUMARATE include BONE DENSITY DECREASED, RENAL INJURY, SKELETAL INJURY, CHRONIC KIDNEY DISEASE, OSTEONECROSIS. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for TENOFOVIR DISOPROXIL FUMARATE.

AI Safety Analysis

Tenofovir Disoproxil Fumarate has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 123,510 adverse event reports for this medication, which is primarily manufactured by Gilead Sciences, Inc..

The most commonly reported adverse events include Bone Density Decreased, Renal Injury, Skeletal Injury. Of classified reports, 94.0% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Bone density decreased and renal injury are the most frequent and serious adverse reactions.

Multiple fractures and chronic kidney disease are also significant concerns. Osteoporosis and osteopenia are common, indicating long-term bone health risks.

Patients taking Tenofovir Disoproxil Fumarate should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Tenofovir disoproxil fumarate can cause bone and renal toxicity, and patients should be monitored for these conditions. Drug interactions, particularly with other nephrotoxic or bone toxic agents, should be avoided. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Tenofovir Disoproxil Fumarate received a safety concern score of 85/100 (high concern). This is based on a 94.0% serious event ratio across 32,657 classified reports. The score accounts for 123,510 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

BONE DENSITY DECREASED10,625 reports
RENAL INJURY9,276 reports
SKELETAL INJURY8,327 reports
CHRONIC KIDNEY DISEASE7,247 reports
OSTEONECROSIS7,245 reports
BONE LOSS7,054 reports
MULTIPLE FRACTURES6,812 reports
RENAL FAILURE6,659 reports
OSTEOPOROSIS5,367 reports
TOOTH LOSS4,498 reports
PAIN3,030 reports
EMOTIONAL DISTRESS2,850 reports
ANXIETY2,668 reports
ANHEDONIA2,451 reports
OSTEOPENIA2,244 reports
TOOTH INJURY2,008 reports
BLOOD CREATININE INCREASED1,631 reports
RENAL IMPAIRMENT1,518 reports
ACUTE KIDNEY INJURY1,199 reports
NEPHROPATHY1,062 reports
FOETAL EXPOSURE DURING PREGNANCY916 reports
DRUG INEFFECTIVE908 reports
ECONOMIC PROBLEM907 reports
VIROLOGIC FAILURE831 reports
PATHOGEN RESISTANCE799 reports
FRACTURE796 reports
DRUG RESISTANCE736 reports
VIRAL MUTATION IDENTIFIED733 reports
DEATH597 reports
FATIGUE583 reports
END STAGE RENAL DISEASE567 reports
FANCONI SYNDROME ACQUIRED557 reports
MATERNAL EXPOSURE DURING PREGNANCY547 reports
DEPRESSION525 reports
NAUSEA524 reports
DRUG INTERACTION508 reports
ANAEMIA504 reports
VITAMIN D DEFICIENCY485 reports
BONE DISORDER478 reports
PYREXIA471 reports
DIARRHOEA465 reports
ASTHENIA449 reports
ABORTION SPONTANEOUS446 reports
PROTEIN TOTAL ABNORMAL446 reports
FOOT FRACTURE436 reports
VOMITING425 reports
OFF LABEL USE423 reports
HEADACHE400 reports
PROTEINURIA397 reports
RASH372 reports
ALANINE AMINOTRANSFERASE INCREASED353 reports
ARTHRALGIA352 reports
TREATMENT FAILURE334 reports
IMMUNE RECONSTITUTION INFLAMMATORY SYNDROME331 reports
RENAL FAILURE ACUTE313 reports
BONE DENSITY ABNORMAL311 reports
EXPOSURE DURING PREGNANCY307 reports
HEPATITIS B303 reports
WEIGHT DECREASED303 reports
OSTEOARTHRITIS300 reports
NEPHROPATHY TOXIC293 reports
TOOTH FRACTURE291 reports
BONE DEMINERALISATION288 reports
ANKLE FRACTURE283 reports
LIPODYSTROPHY ACQUIRED277 reports
CONDITION AGGRAVATED275 reports
RIB FRACTURE273 reports
TREATMENT NONCOMPLIANCE270 reports
GAIT DISTURBANCE268 reports
NEPHROLITHIASIS265 reports
DYSPNOEA263 reports
ASPARTATE AMINOTRANSFERASE INCREASED257 reports
HYPOPHOSPHATAEMIA254 reports
ABDOMINAL PAIN251 reports
DRUG EXPOSURE DURING PREGNANCY244 reports
OSTEOMALACIA244 reports
LOSS OF PERSONAL INDEPENDENCE IN DAILY ACTIVITIES241 reports
BACK PAIN234 reports
HIP FRACTURE229 reports
HYPERTENSION226 reports
VIRAL LOAD INCREASED222 reports
WRIST FRACTURE219 reports
PREMATURE BABY218 reports
DIZZINESS216 reports
MALAISE216 reports
RENAL TUBULAR DISORDER215 reports
HEPATIC FAILURE211 reports
HAND FRACTURE209 reports
BONE PAIN205 reports
GLOMERULAR FILTRATION RATE ABNORMAL204 reports
MITOCHONDRIAL TOXICITY203 reports
RHEUMATOID ARTHRITIS203 reports
DECREASED APPETITE202 reports
HEPATIC CIRRHOSIS202 reports
BLOOD HIV RNA INCREASED193 reports
PAIN IN EXTREMITY190 reports
LACTIC ACIDOSIS188 reports
RENAL DISORDER188 reports
EYELID PTOSIS186 reports
DYSPHAGIA185 reports

Key Safety Signals

  • Bone density decreased and osteoporosis are reported in a significant number of cases.
  • Renal injury and chronic kidney disease are among the top reported adverse reactions.
  • Multiple fractures and osteopenia are also key safety signals.

Patient Demographics

Adverse event reports by sex: Male: 19,216, Female: 9,209, Unknown: 78. The most frequently reported age groups are age 54 (795 reports), age 50 (790 reports), age 52 (692 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 32,657 classified reports for TENOFOVIR DISOPROXIL FUMARATE:

  • Serious: 30,705 reports (94.0%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 1,952 reports (6.0%)
Serious 94.0%Non-Serious 6.0%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male19,216 (67.4%)
Female9,209 (32.3%)
Unknown78 (0.3%)

Reports by Age

Age 54795 reports
Age 50790 reports
Age 52692 reports
Age 51664 reports
Age 55641 reports
Age 53601 reports
Age 48583 reports
Age 49573 reports
Age 47547 reports
Age 44534 reports
Age 46524 reports
Age 45523 reports
Age 57521 reports
Age 56517 reports
Age 43504 reports
Age 41457 reports
Age 59457 reports
Age 40445 reports
Age 39425 reports
Age 42424 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Tenofovir disoproxil fumarate can cause bone and renal toxicity, and patients should be monitored for these conditions. Drug interactions, particularly with other nephrotoxic or bone toxic agents, should be avoided.

What You Should Know

If you are taking Tenofovir Disoproxil Fumarate, here are important things to know. The most commonly reported side effects include bone density decreased, renal injury, skeletal injury, chronic kidney disease, osteonecrosis. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Patients should inform their healthcare provider about any existing bone or kidney conditions before starting Tenofovir disoproxil fumarate. Regular bone density and kidney function tests are recommended during treatment. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA has issued warnings regarding the potential for bone and renal toxicity with Tenofovir disoproxil fumarate. Healthcare providers should closely monitor patients for these adverse events and adjust treatment as necessary.

Frequently Asked Questions

How many adverse event reports has the FDA received for Tenofovir Disoproxil Fumarate?

The FDA has received approximately 123,510 adverse event reports associated with Tenofovir Disoproxil Fumarate. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Tenofovir Disoproxil Fumarate?

The most frequently reported adverse events for Tenofovir Disoproxil Fumarate include Bone Density Decreased, Renal Injury, Skeletal Injury, Chronic Kidney Disease, Osteonecrosis. By volume, the top reported reactions are: Bone Density Decreased (10,625 reports), Renal Injury (9,276 reports), Skeletal Injury (8,327 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Tenofovir Disoproxil Fumarate.

What percentage of Tenofovir Disoproxil Fumarate adverse event reports are serious?

Out of 32,657 classified reports, 30,705 (94.0%) were classified as serious and 1,952 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Tenofovir Disoproxil Fumarate (by sex)?

Adverse event reports for Tenofovir Disoproxil Fumarate break down by patient sex as follows: Male: 19,216, Female: 9,209, Unknown: 78. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Tenofovir Disoproxil Fumarate?

The most frequently reported age groups for Tenofovir Disoproxil Fumarate adverse events are: age 54: 795 reports, age 50: 790 reports, age 52: 692 reports, age 51: 664 reports, age 55: 641 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Tenofovir Disoproxil Fumarate?

The primary manufacturer associated with Tenofovir Disoproxil Fumarate adverse event reports is Gilead Sciences, Inc.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Tenofovir Disoproxil Fumarate?

Beyond the most common reactions, other reported adverse events for Tenofovir Disoproxil Fumarate include: Bone Loss, Multiple Fractures, Renal Failure, Osteoporosis, Tooth Loss. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Tenofovir Disoproxil Fumarate?

You can report adverse events from Tenofovir Disoproxil Fumarate to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Tenofovir Disoproxil Fumarate's safety score and what does it mean?

Tenofovir Disoproxil Fumarate has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Bone density decreased and renal injury are the most frequent and serious adverse reactions.

What are the key safety signals for Tenofovir Disoproxil Fumarate?

Key safety signals identified in Tenofovir Disoproxil Fumarate's adverse event data include: Bone density decreased and osteoporosis are reported in a significant number of cases.. Renal injury and chronic kidney disease are among the top reported adverse reactions.. Multiple fractures and osteopenia are also key safety signals.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Tenofovir Disoproxil Fumarate interact with other drugs?

Tenofovir disoproxil fumarate can cause bone and renal toxicity, and patients should be monitored for these conditions. Drug interactions, particularly with other nephrotoxic or bone toxic agents, should be avoided. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Tenofovir Disoproxil Fumarate.

What should patients know before taking Tenofovir Disoproxil Fumarate?

Patients should inform their healthcare provider about any existing bone or kidney conditions before starting Tenofovir disoproxil fumarate. Regular bone density and kidney function tests are recommended during treatment.

Are Tenofovir Disoproxil Fumarate side effects well-documented?

Tenofovir Disoproxil Fumarate has 123,510 adverse event reports on file with the FDA. Multiple fractures and chronic kidney disease are also significant concerns. The volume of reports for Tenofovir Disoproxil Fumarate reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Tenofovir Disoproxil Fumarate?

The FDA has issued warnings regarding the potential for bone and renal toxicity with Tenofovir disoproxil fumarate. Healthcare providers should closely monitor patients for these adverse events and adjust treatment as necessary. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to TENOFOVIR DISOPROXIL FUMARATE based on therapeutic use, drug class, or shared indications:

EmtricitabineAdefovir dipivoxilEntecavirLamivudineRilpivirine
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.