TRIFLURIDINE AND TIPIRACIL

85/100 · Critical

Manufactured by Taiho Pharmaceutical Co., Ltd.

High Serious Adverse Event Rate for Trifluridine and Tipiracil

21,382 FDA adverse event reports analyzed

Last updated: 2026-05-12

About TRIFLURIDINE AND TIPIRACIL

TRIFLURIDINE AND TIPIRACIL is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Taiho Pharmaceutical Co., Ltd.. Based on analysis of 21,382 FDA adverse event reports, TRIFLURIDINE AND TIPIRACIL has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for TRIFLURIDINE AND TIPIRACIL include DEATH, DISEASE PROGRESSION, FATIGUE, NAUSEA, DIARRHOEA. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for TRIFLURIDINE AND TIPIRACIL.

AI Safety Analysis

Trifluridine And Tipiracil has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 21,382 adverse event reports for this medication, which is primarily manufactured by Taiho Pharmaceutical Co., Ltd..

The most commonly reported adverse events include Death, Disease Progression, Fatigue. Of classified reports, 78.5% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. The drug has a high rate of serious adverse events, including death and disease progression.

Fatigue, nausea, and diarrhea are common side effects reported by patients. There is a significant risk of hematological adverse events, such as decreased white blood cell count and anemia. The drug is associated with a high incidence of gastrointestinal issues, including constipation and abdominal pain.

Patients taking Trifluridine And Tipiracil should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Trifluridine and Tipiracil can cause significant hematological and gastrointestinal side effects, and patients should be monitored closely for these issues. Drug interactions and inappropriate administration schedules are also important to avoid. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Trifluridine And Tipiracil received a safety concern score of 85/100 (high concern). This is based on a 78.5% serious event ratio across 10,345 classified reports. The score accounts for 21,382 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

DEATH3,062 reports
DISEASE PROGRESSION1,779 reports
FATIGUE1,347 reports
NAUSEA1,134 reports
DIARRHOEA970 reports
DECREASED APPETITE658 reports
VOMITING606 reports
WHITE BLOOD CELL COUNT DECREASED479 reports
ASTHENIA471 reports
DRUG INEFFECTIVE358 reports
ANAEMIA345 reports
CONSTIPATION319 reports
WEIGHT DECREASED318 reports
DEHYDRATION311 reports
OFF LABEL USE310 reports
NEUTROPENIA308 reports
ABDOMINAL PAIN307 reports
INAPPROPRIATE SCHEDULE OF PRODUCT ADMINISTRATION296 reports
PAIN257 reports
MALAISE254 reports
ABDOMINAL PAIN UPPER247 reports
PYREXIA244 reports
PLATELET COUNT DECREASED223 reports
DYSPNOEA211 reports
MALIGNANT NEOPLASM PROGRESSION191 reports
HAEMOGLOBIN DECREASED176 reports
CYTOPENIA173 reports
ALOPECIA172 reports
DIZZINESS163 reports
URINARY TRACT INFECTION159 reports
INTESTINAL OBSTRUCTION141 reports
NEUROPATHY PERIPHERAL137 reports
PNEUMONIA137 reports
RED BLOOD CELL COUNT DECREASED137 reports
HEADACHE129 reports
NEUTROPHIL COUNT DECREASED128 reports
HOSPITALISATION124 reports
FALL120 reports
BACK PAIN118 reports
COUGH114 reports
THROMBOCYTOPENIA112 reports
TRANSFUSION104 reports
ASCITES103 reports
HYPOTENSION103 reports
PRODUCT DOSE OMISSION IN ERROR101 reports
ABDOMINAL DISCOMFORT95 reports
STOMATITIS94 reports
HYPERTENSION92 reports
INFECTION92 reports
PAIN IN EXTREMITY92 reports
DYSGEUSIA89 reports
ILLNESS89 reports
INTENTIONAL PRODUCT USE ISSUE89 reports
RASH87 reports
PERIPHERAL SWELLING85 reports
HAEMORRHAGE83 reports
ACUTE KIDNEY INJURY82 reports
SEPSIS80 reports
ABDOMINAL DISTENSION78 reports
ARTHRALGIA78 reports
GENERAL PHYSICAL HEALTH DETERIORATION78 reports
DRUG DOSE OMISSION77 reports
THERAPY INTERRUPTED73 reports
FEBRILE NEUTROPENIA69 reports
INAPPROPRIATE SCHEDULE OF DRUG ADMINISTRATION69 reports
PANCYTOPENIA69 reports
THROMBOSIS69 reports
COLORECTAL CANCER METASTATIC68 reports
PRODUCT USE ISSUE68 reports
LEUKOPENIA67 reports
BLOOD BILIRUBIN INCREASED66 reports
RENAL IMPAIRMENT65 reports
SOMNOLENCE65 reports
GASTROINTESTINAL HAEMORRHAGE64 reports
INSOMNIA64 reports
PRODUCT DOSE OMISSION ISSUE64 reports
JAUNDICE63 reports
BLOOD COUNT ABNORMAL62 reports
CONFUSIONAL STATE62 reports
RECTAL HAEMORRHAGE62 reports
FLATULENCE61 reports
GAIT DISTURBANCE61 reports
HYPOAESTHESIA61 reports
COVID 1958 reports
RENAL FAILURE58 reports
THERAPY CESSATION57 reports
MUSCLE SPASMS56 reports
CHEST PAIN55 reports
FEELING ABNORMAL53 reports
PLEURAL EFFUSION53 reports
HEPATIC FAILURE52 reports
EPISTAXIS51 reports
HAEMATOCHEZIA51 reports
MUSCULAR WEAKNESS51 reports
CARCINOEMBRYONIC ANTIGEN INCREASED50 reports
CEREBROVASCULAR ACCIDENT50 reports
COLON CANCER50 reports
DYSPHONIA50 reports
INCORRECT DOSE ADMINISTERED50 reports
DEEP VEIN THROMBOSIS49 reports

Key Safety Signals

  • Death and disease progression are among the most serious reactions reported.
  • Hematological adverse events, particularly decreased white blood cell count and anemia, are frequent.
  • Gastrointestinal issues, such as constipation and abdominal pain, are commonly reported.
  • There is a notable risk of infections and sepsis.
  • The drug is associated with a high rate of hospitalization and therapy interruption.

Patient Demographics

Adverse event reports by sex: Male: 5,883, Female: 4,255, Unknown: 1. The most frequently reported age groups are age 68 (275 reports), age 66 (262 reports), age 69 (261 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 10,345 classified reports for TRIFLURIDINE AND TIPIRACIL:

  • Serious: 8,125 reports (78.5%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 2,220 reports (21.5%)
Serious 78.5%Non-Serious 21.5%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male5,883 (58.0%)
Female4,255 (42.0%)
Unknown1 (0.0%)

Reports by Age

Age 68275 reports
Age 66262 reports
Age 69261 reports
Age 62258 reports
Age 70254 reports
Age 65250 reports
Age 67246 reports
Age 61231 reports
Age 63224 reports
Age 72219 reports
Age 73218 reports
Age 64217 reports
Age 60213 reports
Age 71209 reports
Age 57203 reports
Age 75200 reports
Age 59198 reports
Age 76187 reports
Age 58186 reports
Age 74184 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Trifluridine and Tipiracil can cause significant hematological and gastrointestinal side effects, and patients should be monitored closely for these issues. Drug interactions and inappropriate administration schedules are also important to avoid.

What You Should Know

If you are taking Trifluridine And Tipiracil, here are important things to know. The most commonly reported side effects include death, disease progression, fatigue, nausea, diarrhoea. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Monitor patients closely for signs of hematological and gastrointestinal side effects, and adjust dosing as necessary. Educate patients on the importance of following the prescribed schedule and dosing instructions. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

Regulatory oversight is ongoing, with the FDA requiring post-marketing surveillance to monitor the drug's safety profile. Patients should report any adverse reactions to their healthcare provider immediately.

Frequently Asked Questions

How many adverse event reports has the FDA received for Trifluridine And Tipiracil?

The FDA has received approximately 21,382 adverse event reports associated with Trifluridine And Tipiracil. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Trifluridine And Tipiracil?

The most frequently reported adverse events for Trifluridine And Tipiracil include Death, Disease Progression, Fatigue, Nausea, Diarrhoea. By volume, the top reported reactions are: Death (3,062 reports), Disease Progression (1,779 reports), Fatigue (1,347 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Trifluridine And Tipiracil.

What percentage of Trifluridine And Tipiracil adverse event reports are serious?

Out of 10,345 classified reports, 8,125 (78.5%) were classified as serious and 2,220 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Trifluridine And Tipiracil (by sex)?

Adverse event reports for Trifluridine And Tipiracil break down by patient sex as follows: Male: 5,883, Female: 4,255, Unknown: 1. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Trifluridine And Tipiracil?

The most frequently reported age groups for Trifluridine And Tipiracil adverse events are: age 68: 275 reports, age 66: 262 reports, age 69: 261 reports, age 62: 258 reports, age 70: 254 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Trifluridine And Tipiracil?

The primary manufacturer associated with Trifluridine And Tipiracil adverse event reports is Taiho Pharmaceutical Co., Ltd.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Trifluridine And Tipiracil?

Beyond the most common reactions, other reported adverse events for Trifluridine And Tipiracil include: Decreased Appetite, Vomiting, White Blood Cell Count Decreased, Asthenia, Drug Ineffective. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Trifluridine And Tipiracil?

You can report adverse events from Trifluridine And Tipiracil to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Trifluridine And Tipiracil's safety score and what does it mean?

Trifluridine And Tipiracil has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. The drug has a high rate of serious adverse events, including death and disease progression.

What are the key safety signals for Trifluridine And Tipiracil?

Key safety signals identified in Trifluridine And Tipiracil's adverse event data include: Death and disease progression are among the most serious reactions reported.. Hematological adverse events, particularly decreased white blood cell count and anemia, are frequent.. Gastrointestinal issues, such as constipation and abdominal pain, are commonly reported.. There is a notable risk of infections and sepsis.. The drug is associated with a high rate of hospitalization and therapy interruption.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Trifluridine And Tipiracil interact with other drugs?

Trifluridine and Tipiracil can cause significant hematological and gastrointestinal side effects, and patients should be monitored closely for these issues. Drug interactions and inappropriate administration schedules are also important to avoid. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Trifluridine And Tipiracil.

What should patients know before taking Trifluridine And Tipiracil?

Monitor patients closely for signs of hematological and gastrointestinal side effects, and adjust dosing as necessary. Educate patients on the importance of following the prescribed schedule and dosing instructions.

Are Trifluridine And Tipiracil side effects well-documented?

Trifluridine And Tipiracil has 21,382 adverse event reports on file with the FDA. Fatigue, nausea, and diarrhea are common side effects reported by patients. The volume of reports for Trifluridine And Tipiracil reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Trifluridine And Tipiracil?

Regulatory oversight is ongoing, with the FDA requiring post-marketing surveillance to monitor the drug's safety profile. Patients should report any adverse reactions to their healthcare provider immediately. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to TRIFLURIDINE AND TIPIRACIL based on therapeutic use, drug class, or shared indications:

TrifluridineTipiracilPemetrexedCisplatinFluorouracil
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.