ENZALUTAMIDE

82/100 · Critical

Manufactured by Astellas Pharma US, Inc.

Enzalutamide Adverse Events: High Serious Reaction Rate

117,902 FDA adverse event reports analyzed

Last updated: 2026-05-12

About ENZALUTAMIDE

ENZALUTAMIDE is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Astellas Pharma US, Inc.. Based on analysis of 117,902 FDA adverse event reports, ENZALUTAMIDE has a safety score of 82 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for ENZALUTAMIDE include FATIGUE, DEATH, MALIGNANT NEOPLASM PROGRESSION, PROSTATIC SPECIFIC ANTIGEN INCREASED, ASTHENIA. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for ENZALUTAMIDE.

AI Safety Analysis

Enzalutamide has a safety concern score of 82 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 117,902 adverse event reports for this medication, which is primarily manufactured by Astellas Pharma Us, Inc..

The most commonly reported adverse events include Fatigue, Death, Malignant Neoplasm Progression. Of classified reports, 61.4% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Fatigue and asthenia are the most common adverse events, with over 10,000 reports each.

Serious adverse events, including death and malignant neoplasm progression, account for 61.4% of all reports. The most frequent serious reactions include death, malignant neoplasm progression, and heart-related issues.

Patients taking Enzalutamide should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Enzalutamide can interact with other drugs, leading to adverse effects. Patients should inform their healthcare providers of all medications they are taking. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 82/100

Enzalutamide received a safety concern score of 82/100 (high concern). This is based on a 61.4% serious event ratio across 57,602 classified reports. The score accounts for 117,902 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

FATIGUE10,159 reports
DEATH7,667 reports
MALIGNANT NEOPLASM PROGRESSION5,409 reports
PROSTATIC SPECIFIC ANTIGEN INCREASED4,295 reports
ASTHENIA4,120 reports
DRUG INEFFECTIVE4,028 reports
HOT FLUSH3,819 reports
DECREASED APPETITE3,379 reports
NAUSEA3,240 reports
DIZZINESS3,107 reports
DIARRHOEA2,783 reports
BACK PAIN2,282 reports
ARTHRALGIA2,124 reports
UNDERDOSE2,067 reports
CONSTIPATION1,807 reports
FALL1,790 reports
WEIGHT DECREASED1,777 reports
PAIN1,708 reports
HEADACHE1,650 reports
MALAISE1,559 reports
DYSPNOEA1,483 reports
INSOMNIA1,354 reports
PERIPHERAL SWELLING1,316 reports
DYSPHAGIA1,296 reports
VOMITING1,255 reports
PAIN IN EXTREMITY1,215 reports
OFF LABEL USE1,024 reports
SOMNOLENCE1,007 reports
MUSCULAR WEAKNESS1,001 reports
ABDOMINAL DISCOMFORT983 reports
MYALGIA957 reports
DRUG DOSE OMISSION937 reports
CONFUSIONAL STATE914 reports
DRUG INTERACTION881 reports
GAIT DISTURBANCE848 reports
ANAEMIA846 reports
PROSTATE CANCER839 reports
FEELING ABNORMAL835 reports
RASH827 reports
MEMORY IMPAIRMENT814 reports
BONE PAIN789 reports
URINARY TRACT INFECTION765 reports
BLOOD PRESSURE INCREASED736 reports
PNEUMONIA723 reports
HYPERTENSION721 reports
BALANCE DISORDER689 reports
CEREBROVASCULAR ACCIDENT651 reports
HYPERHIDROSIS644 reports
NEUROPATHY PERIPHERAL630 reports
HYPOAESTHESIA618 reports
TREATMENT NONCOMPLIANCE611 reports
PRODUCT SIZE ISSUE606 reports
DYSGEUSIA605 reports
ABDOMINAL PAIN UPPER582 reports
ANXIETY574 reports
PRURITUS571 reports
GENERAL PHYSICAL HEALTH DETERIORATION564 reports
DEPRESSION545 reports
DEHYDRATION541 reports
PARAESTHESIA541 reports
METASTASES TO BONE533 reports
SEIZURE510 reports
OEDEMA PERIPHERAL504 reports
WEIGHT INCREASED499 reports
VISION BLURRED494 reports
HOSPITALISATION487 reports
PYREXIA482 reports
COUGH479 reports
LOSS OF CONSCIOUSNESS472 reports
MUSCLE SPASMS469 reports
AMNESIA460 reports
CHEST PAIN456 reports
POLLAKIURIA438 reports
CONDITION AGGRAVATED414 reports
MYOCARDIAL INFARCTION408 reports
PRODUCT STORAGE ERROR408 reports
JOINT SWELLING402 reports
NASOPHARYNGITIS392 reports
HAEMOGLOBIN DECREASED391 reports
TREMOR386 reports
CARDIAC FAILURE384 reports
INAPPROPRIATE SCHEDULE OF DRUG ADMINISTRATION376 reports
MUSCULOSKELETAL PAIN370 reports
DISEASE PROGRESSION358 reports
HYPOTENSION353 reports
ATRIAL FIBRILLATION351 reports
ABDOMINAL PAIN348 reports
HALLUCINATION348 reports
ALOPECIA346 reports
PRODUCT USE COMPLAINT343 reports
LETHARGY334 reports
BLOOD URINE PRESENT329 reports
VISUAL IMPAIRMENT327 reports
INCORRECT DOSE ADMINISTERED325 reports
HAEMATURIA313 reports
PROSTATE CANCER METASTATIC306 reports
PRODUCT DOSE OMISSION303 reports
DRUG INTOLERANCE300 reports
DYSPEPSIA298 reports
PLATELET COUNT DECREASED298 reports

Key Safety Signals

  • Death and malignant neoplasm progression are the most critical safety signals.
  • Heart-related issues, including myocardial infarction and atrial fibrillation, are also significant.
  • Drug ineffectiveness and underdose are common, indicating potential dosing issues.

Patient Demographics

Adverse event reports by sex: Male: 54,925, Female: 361, Unknown: 83. The most frequently reported age groups are age 78 (1,378 reports), age 75 (1,320 reports), age 79 (1,309 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 57,602 classified reports for ENZALUTAMIDE:

  • Serious: 35,395 reports (61.4%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 22,207 reports (38.6%)
Serious 61.4%Non-Serious 38.6%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male54,925 (99.2%)
Female361 (0.7%)
Unknown83 (0.1%)

Reports by Age

Age 781,378 reports
Age 751,320 reports
Age 791,309 reports
Age 771,293 reports
Age 741,264 reports
Age 801,258 reports
Age 761,224 reports
Age 731,195 reports
Age 821,185 reports
Age 721,175 reports
Age 811,170 reports
Age 831,159 reports
Age 711,124 reports
Age 701,093 reports
Age 841,072 reports
Age 851,001 reports
Age 86944 reports
Age 69935 reports
Age 67924 reports
Age 68879 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Enzalutamide can interact with other drugs, leading to adverse effects. Patients should inform their healthcare providers of all medications they are taking.

What You Should Know

If you are taking Enzalutamide, here are important things to know. The most commonly reported side effects include fatigue, death, malignant neoplasm progression, prostatic specific antigen increased, asthenia. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Monitor for signs of fatigue and weakness, which are common and can be severe. Report any serious adverse events immediately to your healthcare provider. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

Regulatory oversight is ongoing, with the FDA requiring post-marketing studies to further evaluate long-term safety and efficacy.

Frequently Asked Questions

How many adverse event reports has the FDA received for Enzalutamide?

The FDA has received approximately 117,902 adverse event reports associated with Enzalutamide. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Enzalutamide?

The most frequently reported adverse events for Enzalutamide include Fatigue, Death, Malignant Neoplasm Progression, Prostatic Specific Antigen Increased, Asthenia. By volume, the top reported reactions are: Fatigue (10,159 reports), Death (7,667 reports), Malignant Neoplasm Progression (5,409 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Enzalutamide.

What percentage of Enzalutamide adverse event reports are serious?

Out of 57,602 classified reports, 35,395 (61.4%) were classified as serious and 22,207 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Enzalutamide (by sex)?

Adverse event reports for Enzalutamide break down by patient sex as follows: Male: 54,925, Female: 361, Unknown: 83. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Enzalutamide?

The most frequently reported age groups for Enzalutamide adverse events are: age 78: 1,378 reports, age 75: 1,320 reports, age 79: 1,309 reports, age 77: 1,293 reports, age 74: 1,264 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Enzalutamide?

The primary manufacturer associated with Enzalutamide adverse event reports is Astellas Pharma Us, Inc.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Enzalutamide?

Beyond the most common reactions, other reported adverse events for Enzalutamide include: Drug Ineffective, Hot Flush, Decreased Appetite, Nausea, Dizziness. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Enzalutamide?

You can report adverse events from Enzalutamide to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Enzalutamide's safety score and what does it mean?

Enzalutamide has a safety concern score of 82 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Fatigue and asthenia are the most common adverse events, with over 10,000 reports each.

What are the key safety signals for Enzalutamide?

Key safety signals identified in Enzalutamide's adverse event data include: Death and malignant neoplasm progression are the most critical safety signals.. Heart-related issues, including myocardial infarction and atrial fibrillation, are also significant.. Drug ineffectiveness and underdose are common, indicating potential dosing issues.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Enzalutamide interact with other drugs?

Enzalutamide can interact with other drugs, leading to adverse effects. Patients should inform their healthcare providers of all medications they are taking. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Enzalutamide.

What should patients know before taking Enzalutamide?

Monitor for signs of fatigue and weakness, which are common and can be severe. Report any serious adverse events immediately to your healthcare provider.

Are Enzalutamide side effects well-documented?

Enzalutamide has 117,902 adverse event reports on file with the FDA. Serious adverse events, including death and malignant neoplasm progression, account for 61.4% of all reports. The volume of reports for Enzalutamide reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Enzalutamide?

Regulatory oversight is ongoing, with the FDA requiring post-marketing studies to further evaluate long-term safety and efficacy. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to ENZALUTAMIDE based on therapeutic use, drug class, or shared indications:

WarfarinDigoxinCimetidine
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.