TACROLIMUS EXTENDED RELEASE CAPSULES

85/100 · Critical

Manufactured by Astellas Pharma US, Inc.

High Safety Concerns with Tacrolimus Extended-Release Capsules

181,869 FDA adverse event reports analyzed

Last updated: 2026-05-12

About TACROLIMUS EXTENDED RELEASE CAPSULES

TACROLIMUS EXTENDED RELEASE CAPSULES is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Astellas Pharma US, Inc.. Based on analysis of 181,869 FDA adverse event reports, TACROLIMUS EXTENDED RELEASE CAPSULES has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for TACROLIMUS EXTENDED RELEASE CAPSULES include OFF LABEL USE, DRUG INEFFECTIVE, PRODUCT USE IN UNAPPROVED INDICATION, DRUG INTERACTION, ACUTE KIDNEY INJURY. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for TACROLIMUS EXTENDED RELEASE CAPSULES.

AI Safety Analysis

Tacrolimus Extended-Release Capsules has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 181,869 adverse event reports for this medication, which is primarily manufactured by Astellas Pharma Us, Inc..

The most commonly reported adverse events include Off Label Use, Drug Ineffective, Product Use In Unapproved Indication. Of classified reports, 90.7% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Acute kidney injury and renal impairment are among the most serious adverse events reported.

Drug interactions and ineffective drug performance are common issues. Infections, particularly cytomegalovirus and pneumonia, are frequent and serious.

Patients taking Tacrolimus Extended-Release Capsules should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Tacrolimus can interact with various drugs, potentially leading to increased toxicity or reduced efficacy. Warnings are issued for specific drug combinations. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Tacrolimus Extended-Release Capsules received a safety concern score of 85/100 (high concern). This is based on a 90.7% serious event ratio across 117,850 classified reports. The score accounts for 181,869 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

OFF LABEL USE11,734 reports
DRUG INEFFECTIVE8,329 reports
PRODUCT USE IN UNAPPROVED INDICATION5,813 reports
DRUG INTERACTION5,363 reports
ACUTE KIDNEY INJURY5,057 reports
DIARRHOEA4,324 reports
TRANSPLANT REJECTION3,983 reports
CYTOMEGALOVIRUS INFECTION3,844 reports
PYREXIA3,690 reports
COVID 193,632 reports
TOXICITY TO VARIOUS AGENTS3,493 reports
PNEUMONIA3,351 reports
DEATH3,291 reports
RENAL IMPAIRMENT2,734 reports
SEPSIS2,712 reports
POST TRANSPLANT LYMPHOPROLIFERATIVE DISORDER2,699 reports
CONDITION AGGRAVATED2,503 reports
NAUSEA2,335 reports
THROMBOTIC MICROANGIOPATHY2,296 reports
RESPIRATORY FAILURE2,261 reports
ANAEMIA2,158 reports
BLOOD CREATININE INCREASED2,117 reports
VOMITING2,096 reports
SEPTIC SHOCK2,042 reports
MULTIPLE ORGAN DYSFUNCTION SYNDROME2,030 reports
RENAL FAILURE1,991 reports
URINARY TRACT INFECTION1,935 reports
NEUTROPENIA1,908 reports
DYSPNOEA1,853 reports
HEADACHE1,841 reports
LEUKOPENIA1,825 reports
INFECTION1,819 reports
IMMUNOSUPPRESSANT DRUG LEVEL INCREASED1,786 reports
FATIGUE1,785 reports
HYPERTENSION1,741 reports
RASH1,698 reports
KIDNEY TRANSPLANT REJECTION1,696 reports
THROMBOCYTOPENIA1,642 reports
PANCYTOPENIA1,612 reports
POLYOMAVIRUS ASSOCIATED NEPHROPATHY1,611 reports
CYTOMEGALOVIRUS VIRAEMIA1,549 reports
DRUG LEVEL INCREASED1,495 reports
PRURITUS1,494 reports
ABDOMINAL PAIN1,459 reports
EPSTEIN BARR VIRUS INFECTION1,415 reports
DRUG INEFFECTIVE FOR UNAPPROVED INDICATION1,401 reports
GRAFT VERSUS HOST DISEASE1,389 reports
BK VIRUS INFECTION1,342 reports
WEIGHT DECREASED1,271 reports
POSTERIOR REVERSIBLE ENCEPHALOPATHY SYNDROME1,209 reports
ASPERGILLUS INFECTION1,185 reports
BRONCHOPULMONARY ASPERGILLOSIS1,182 reports
NEPHROPATHY TOXIC1,172 reports
ASTHENIA1,162 reports
COUGH1,156 reports
PAIN1,155 reports
FEBRILE NEUTROPENIA1,134 reports
PNEUMOCYSTIS JIROVECII PNEUMONIA1,118 reports
TREMOR1,113 reports
CYTOMEGALOVIRUS INFECTION REACTIVATION1,063 reports
PLEURAL EFFUSION1,056 reports
CHRONIC KIDNEY DISEASE1,051 reports
ACUTE GRAFT VERSUS HOST DISEASE1,049 reports
PRODUCT USE ISSUE1,046 reports
HYPOTENSION1,041 reports
COMPLICATIONS OF TRANSPLANTED KIDNEY1,027 reports
TREATMENT FAILURE1,027 reports
DIABETES MELLITUS1,025 reports
MALAISE1,025 reports
DISEASE PROGRESSION993 reports
DISEASE RECURRENCE964 reports
ACUTE RESPIRATORY DISTRESS SYNDROME961 reports
STAPHYLOCOCCAL INFECTION946 reports
CHRONIC GRAFT VERSUS HOST DISEASE923 reports
MATERNAL EXPOSURE DURING PREGNANCY921 reports
DECREASED APPETITE915 reports
NOCARDIOSIS906 reports
HYPERKALAEMIA902 reports
FUNGAL INFECTION897 reports
FOETAL EXPOSURE DURING PREGNANCY876 reports
EXPOSURE DURING PREGNANCY870 reports
KLEBSIELLA INFECTION870 reports
ARTHRALGIA866 reports
DRUG RESISTANCE858 reports
TRANSPLANT DYSFUNCTION856 reports
PSEUDOMONAS INFECTION853 reports
ENTEROCOCCAL INFECTION833 reports
HAEMOGLOBIN DECREASED831 reports
DERMATITIS ATOPIC814 reports
ESCHERICHIA INFECTION811 reports
ADENOVIRUS INFECTION807 reports
NEUROTOXICITY806 reports
KAPOSI^S SARCOMA795 reports
ERYTHEMA791 reports
ACUTE GRAFT VERSUS HOST DISEASE IN SKIN770 reports
PROTEINURIA766 reports
DEHYDRATION763 reports
BACTERAEMIA760 reports
DRUG INTOLERANCE753 reports
PREMATURE BABY751 reports

Key Safety Signals

  • Acute kidney injury and renal impairment
  • Drug interactions and ineffectiveness
  • Frequent and serious infections

Patient Demographics

Adverse event reports by sex: Male: 57,391, Female: 43,746, Unknown: 605. The most frequently reported age groups are age 57 (2,140 reports), age 58 (2,101 reports), age 55 (2,052 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 117,850 classified reports for TACROLIMUS EXTENDED RELEASE CAPSULES:

  • Serious: 106,867 reports (90.7%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 10,983 reports (9.3%)
Serious 90.7%Non-Serious 9.3%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male57,391 (56.4%)
Female43,746 (43.0%)
Unknown605 (0.6%)

Reports by Age

Age 572,140 reports
Age 582,101 reports
Age 552,052 reports
Age 592,050 reports
Age 652,035 reports
Age 602,027 reports
Age 632,024 reports
Age 611,978 reports
Age 641,972 reports
Age 621,941 reports
Age 561,892 reports
Age 681,795 reports
Age 521,770 reports
Age 671,746 reports
Age 661,735 reports
Age 511,682 reports
Age 541,680 reports
Age 531,678 reports
Age 501,674 reports
Age 691,557 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Tacrolimus can interact with various drugs, potentially leading to increased toxicity or reduced efficacy. Warnings are issued for specific drug combinations.

What You Should Know

If you are taking Tacrolimus Extended-Release Capsules, here are important things to know. The most commonly reported side effects include off label use, drug ineffective, product use in unapproved indication, drug interaction, acute kidney injury. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Monitor kidney function regularly, especially in patients with pre-existing kidney conditions. Be cautious with drug interactions and inform healthcare providers of all medications being taken. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA closely monitors Tacrolimus Extended-Release Capsules due to high safety concerns, particularly for kidney function and infections.

Frequently Asked Questions

How many adverse event reports has the FDA received for Tacrolimus Extended-Release Capsules?

The FDA has received approximately 181,869 adverse event reports associated with Tacrolimus Extended-Release Capsules. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Tacrolimus Extended-Release Capsules?

The most frequently reported adverse events for Tacrolimus Extended-Release Capsules include Off Label Use, Drug Ineffective, Product Use In Unapproved Indication, Drug Interaction, Acute Kidney Injury. By volume, the top reported reactions are: Off Label Use (11,734 reports), Drug Ineffective (8,329 reports), Product Use In Unapproved Indication (5,813 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Tacrolimus Extended-Release Capsules.

What percentage of Tacrolimus Extended-Release Capsules adverse event reports are serious?

Out of 117,850 classified reports, 106,867 (90.7%) were classified as serious and 10,983 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Tacrolimus Extended-Release Capsules (by sex)?

Adverse event reports for Tacrolimus Extended-Release Capsules break down by patient sex as follows: Male: 57,391, Female: 43,746, Unknown: 605. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Tacrolimus Extended-Release Capsules?

The most frequently reported age groups for Tacrolimus Extended-Release Capsules adverse events are: age 57: 2,140 reports, age 58: 2,101 reports, age 55: 2,052 reports, age 59: 2,050 reports, age 65: 2,035 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Tacrolimus Extended-Release Capsules?

The primary manufacturer associated with Tacrolimus Extended-Release Capsules adverse event reports is Astellas Pharma Us, Inc.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Tacrolimus Extended-Release Capsules?

Beyond the most common reactions, other reported adverse events for Tacrolimus Extended-Release Capsules include: Diarrhoea, Transplant Rejection, Cytomegalovirus Infection, Pyrexia, Covid-19. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Tacrolimus Extended-Release Capsules?

You can report adverse events from Tacrolimus Extended-Release Capsules to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Tacrolimus Extended-Release Capsules's safety score and what does it mean?

Tacrolimus Extended-Release Capsules has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Acute kidney injury and renal impairment are among the most serious adverse events reported.

What are the key safety signals for Tacrolimus Extended-Release Capsules?

Key safety signals identified in Tacrolimus Extended-Release Capsules's adverse event data include: Acute kidney injury and renal impairment. Drug interactions and ineffectiveness. Frequent and serious infections. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Tacrolimus Extended-Release Capsules interact with other drugs?

Tacrolimus can interact with various drugs, potentially leading to increased toxicity or reduced efficacy. Warnings are issued for specific drug combinations. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Tacrolimus Extended-Release Capsules.

What should patients know before taking Tacrolimus Extended-Release Capsules?

Monitor kidney function regularly, especially in patients with pre-existing kidney conditions. Be cautious with drug interactions and inform healthcare providers of all medications being taken.

Are Tacrolimus Extended-Release Capsules side effects well-documented?

Tacrolimus Extended-Release Capsules has 181,869 adverse event reports on file with the FDA. Drug interactions and ineffective drug performance are common issues. The volume of reports for Tacrolimus Extended-Release Capsules reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Tacrolimus Extended-Release Capsules?

The FDA closely monitors Tacrolimus Extended-Release Capsules due to high safety concerns, particularly for kidney function and infections. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to TACROLIMUS EXTENDED RELEASE CAPSULES based on therapeutic use, drug class, or shared indications:

CyclosporinePrednisoneMycophenolate mofetil
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.