ESTRADIOL

65/100 · Elevated

Manufactured by Allergan, Inc.

Estradiol Adverse Events: Moderate Safety Concerns

159,657 FDA adverse event reports analyzed

Last updated: 2026-05-12

About ESTRADIOL

ESTRADIOL is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Allergan, Inc.. Based on analysis of 159,657 FDA adverse event reports, ESTRADIOL has a safety score of 65 out of 100. This moderate score indicates a notable volume of adverse event reports that patients and providers should be aware of. The most commonly reported adverse reactions for ESTRADIOL include DRUG INEFFECTIVE, OFF LABEL USE, PRODUCT ADHESION ISSUE, HEADACHE, NAUSEA. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for ESTRADIOL.

AI Safety Analysis

Estradiol has a safety concern score of 65 out of 100, placing it in the elevated concern category based on analysis of FDA adverse event data. The FDA has received approximately 159,657 adverse event reports for this medication, which is primarily manufactured by Allergan, Inc..

The most commonly reported adverse events include Drug Ineffective, Off Label Use, Product Adhesion Issue. Of classified reports, 43.7% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Headache and nausea are the most common adverse events reported.

Serious adverse events account for 43.7% of all reports. The majority of reports are from female patients, with the highest number of reports from patients aged 56-60.

Patients taking Estradiol should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Estradiol can interact with other medications, and patients should be aware of potential drug interactions and follow the prescribed usage instructions. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 65/100

Estradiol received a safety concern score of 65/100 (elevated concern). This is based on a 43.7% serious event ratio across 83,666 classified reports. The score accounts for 159,657 total adverse event reports and 100 distinct reaction types. This elevated score indicates a notable proportion of serious adverse events and warrants careful monitoring.

Top Adverse Reactions

DRUG INEFFECTIVE7,618 reports
OFF LABEL USE5,559 reports
PRODUCT ADHESION ISSUE5,172 reports
HEADACHE5,035 reports
NAUSEA4,753 reports
FATIGUE4,512 reports
PAIN3,478 reports
HOT FLUSH3,279 reports
DIARRHOEA3,055 reports
DIZZINESS2,921 reports
ARTHRALGIA2,820 reports
RASH2,503 reports
DYSPNOEA2,440 reports
BREAST CANCER FEMALE2,438 reports
PRURITUS2,433 reports
PRODUCT QUALITY ISSUE2,425 reports
INSOMNIA2,414 reports
MALAISE2,325 reports
WRONG TECHNIQUE IN PRODUCT USAGE PROCESS2,199 reports
ANXIETY2,150 reports
FEELING ABNORMAL2,100 reports
VOMITING2,083 reports
NO ADVERSE EVENT2,081 reports
PAIN IN EXTREMITY1,924 reports
BREAST CANCER1,875 reports
WEIGHT INCREASED1,802 reports
DEPRESSION1,798 reports
ASTHENIA1,741 reports
BACK PAIN1,661 reports
FALL1,639 reports
ALOPECIA1,636 reports
WEIGHT DECREASED1,590 reports
URINARY TRACT INFECTION1,571 reports
MUSCLE SPASMS1,508 reports
APPLICATION SITE ERYTHEMA1,480 reports
PRODUCT DOSE OMISSION ISSUE1,462 reports
CONDITION AGGRAVATED1,458 reports
APPLICATION SITE PRURITUS1,442 reports
MIGRAINE1,424 reports
COUGH1,410 reports
ABDOMINAL PAIN1,358 reports
PRODUCT USE ISSUE1,275 reports
HYPERSENSITIVITY1,261 reports
CONSTIPATION1,213 reports
APPLICATION SITE RASH1,202 reports
SINUSITIS1,191 reports
ABDOMINAL PAIN UPPER1,189 reports
DRUG HYPERSENSITIVITY1,184 reports
PYREXIA1,163 reports
PNEUMONIA1,153 reports
HYPERTENSION1,140 reports
PARAESTHESIA1,115 reports
HYPERHIDROSIS1,095 reports
INCORRECT DOSE ADMINISTERED1,090 reports
BLOOD PRESSURE INCREASED1,075 reports
URTICARIA1,075 reports
PRODUCT USE IN UNAPPROVED INDICATION1,069 reports
CHEST PAIN1,061 reports
GAIT DISTURBANCE1,054 reports
PALPITATIONS1,044 reports
ABDOMINAL DISCOMFORT1,043 reports
ABDOMINAL DISTENSION1,043 reports
PERIPHERAL SWELLING1,041 reports
INJECTION SITE PAIN1,032 reports
NASOPHARYNGITIS1,032 reports
VAGINAL HAEMORRHAGE1,022 reports
COVID 191,019 reports
MYALGIA998 reports
DEVICE ADHESION ISSUE990 reports
ERYTHEMA962 reports
PRODUCT SUBSTITUTION ISSUE937 reports
HYPOAESTHESIA932 reports
VULVOVAGINAL DISCOMFORT902 reports
TREMOR893 reports
SOMNOLENCE881 reports
MEMORY IMPAIRMENT873 reports
VISION BLURRED856 reports
DECREASED APPETITE835 reports
JOINT SWELLING834 reports
DRUG DOSE OMISSION820 reports
ARTHRITIS809 reports
BRONCHITIS808 reports
INAPPROPRIATE SCHEDULE OF PRODUCT ADMINISTRATION802 reports
NIGHT SWEATS802 reports
APPLICATION SITE IRRITATION791 reports
DRUG INTERACTION778 reports
GASTROOESOPHAGEAL REFLUX DISEASE763 reports
VULVOVAGINAL BURNING SENSATION758 reports
VAGINAL DISCHARGE756 reports
INFECTION727 reports
CONTUSION709 reports
RHEUMATOID ARTHRITIS688 reports
DYSPEPSIA680 reports
CHEST DISCOMFORT671 reports
APPLICATION SITE PAIN666 reports
BURNING SENSATION663 reports
OEDEMA PERIPHERAL659 reports
ANAEMIA658 reports
ASTHMA652 reports
HEART RATE INCREASED651 reports

Key Safety Signals

  • Headache and nausea are the most frequently reported adverse events.
  • Serious adverse events, such as breast cancer and pneumonia, are reported but at lower frequencies.
  • A significant number of reports involve product quality and usage issues.

Patient Demographics

Adverse event reports by sex: Female: 76,888, Male: 1,037, Unknown: 164. The most frequently reported age groups are age 56 (1,586 reports), age 55 (1,582 reports), age 60 (1,569 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 83,666 classified reports for ESTRADIOL:

  • Serious: 36,561 reports (43.7%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 47,105 reports (56.3%)
Serious 43.7%Non-Serious 56.3%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female76,888 (98.5%)
Male1,037 (1.3%)
Unknown164 (0.2%)

Reports by Age

Age 561,586 reports
Age 551,582 reports
Age 601,569 reports
Age 581,564 reports
Age 571,558 reports
Age 591,555 reports
Age 531,506 reports
Age 541,485 reports
Age 621,428 reports
Age 611,404 reports
Age 631,374 reports
Age 641,342 reports
Age 521,315 reports
Age 511,302 reports
Age 651,205 reports
Age 501,156 reports
Age 661,103 reports
Age 671,101 reports
Age 681,050 reports
Age 691,035 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Estradiol can interact with other medications, and patients should be aware of potential drug interactions and follow the prescribed usage instructions.

What You Should Know

If you are taking Estradiol, here are important things to know. The most commonly reported side effects include drug ineffective, off label use, product adhesion issue, headache, nausea. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Follow the prescribed usage instructions carefully to minimize the risk of adverse events. Report any serious adverse events to your healthcare provider immediately. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA continues to monitor the safety of estradiol and may require additional studies or changes to labeling based on ongoing data.

Frequently Asked Questions

How many adverse event reports has the FDA received for Estradiol?

The FDA has received approximately 159,657 adverse event reports associated with Estradiol. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Estradiol?

The most frequently reported adverse events for Estradiol include Drug Ineffective, Off Label Use, Product Adhesion Issue, Headache, Nausea. By volume, the top reported reactions are: Drug Ineffective (7,618 reports), Off Label Use (5,559 reports), Product Adhesion Issue (5,172 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Estradiol.

What percentage of Estradiol adverse event reports are serious?

Out of 83,666 classified reports, 36,561 (43.7%) were classified as serious and 47,105 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Estradiol (by sex)?

Adverse event reports for Estradiol break down by patient sex as follows: Female: 76,888, Male: 1,037, Unknown: 164. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Estradiol?

The most frequently reported age groups for Estradiol adverse events are: age 56: 1,586 reports, age 55: 1,582 reports, age 60: 1,569 reports, age 58: 1,564 reports, age 57: 1,558 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Estradiol?

The primary manufacturer associated with Estradiol adverse event reports is Allergan, Inc.. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Estradiol?

Beyond the most common reactions, other reported adverse events for Estradiol include: Fatigue, Pain, Hot Flush, Diarrhoea, Dizziness. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Estradiol?

You can report adverse events from Estradiol to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Estradiol's safety score and what does it mean?

Estradiol has a safety concern score of 65 out of 100 (elevated concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Headache and nausea are the most common adverse events reported.

What are the key safety signals for Estradiol?

Key safety signals identified in Estradiol's adverse event data include: Headache and nausea are the most frequently reported adverse events.. Serious adverse events, such as breast cancer and pneumonia, are reported but at lower frequencies.. A significant number of reports involve product quality and usage issues.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Estradiol interact with other drugs?

Estradiol can interact with other medications, and patients should be aware of potential drug interactions and follow the prescribed usage instructions. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Estradiol.

What should patients know before taking Estradiol?

Follow the prescribed usage instructions carefully to minimize the risk of adverse events. Report any serious adverse events to your healthcare provider immediately.

Are Estradiol side effects well-documented?

Estradiol has 159,657 adverse event reports on file with the FDA. Serious adverse events account for 43.7% of all reports. The volume of reports for Estradiol reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Estradiol?

The FDA continues to monitor the safety of estradiol and may require additional studies or changes to labeling based on ongoing data. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to ESTRADIOL based on therapeutic use, drug class, or shared indications:

IbuprofenParacetamolAspirin
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.