ESTRADIOL TRANSDERMAL

65/100 · Elevated

Manufactured by Amneal Pharmaceuticals NY LLC

Moderate Safety Concerns with Estradiol Transdermal

79,078 FDA adverse event reports analyzed

Last updated: 2026-05-12

About ESTRADIOL TRANSDERMAL

ESTRADIOL TRANSDERMAL is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Amneal Pharmaceuticals NY LLC. Based on analysis of 79,078 FDA adverse event reports, ESTRADIOL TRANSDERMAL has a safety score of 65 out of 100. This moderate score indicates a notable volume of adverse event reports that patients and providers should be aware of. The most commonly reported adverse reactions for ESTRADIOL TRANSDERMAL include DRUG INEFFECTIVE, NAUSEA, FATIGUE, HEADACHE, OFF LABEL USE. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for ESTRADIOL TRANSDERMAL.

AI Safety Analysis

Estradiol Transdermal has a safety concern score of 65 out of 100, placing it in the elevated concern category based on analysis of FDA adverse event data. The FDA has received approximately 79,078 adverse event reports for this medication, which is primarily manufactured by Amneal Pharmaceuticals Ny Llc.

The most commonly reported adverse events include Drug Ineffective, Nausea, Fatigue. Of classified reports, 49.8% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. The most common reactions include nausea, fatigue, and headache, indicating a broad range of mild to moderate side effects.

Serious adverse events, such as breast cancer and dizziness, are reported but at a lower frequency compared to non-serious events. There is a notable number of drug interaction reports, suggesting potential risks when combined with other medications. The majority of reports are from female patients, which aligns with the drug's intended use for hormone replacement therapy.

Patients taking Estradiol Transdermal should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Drug interactions are a key safety signal, with 575 reports indicating potential risks when combined with other medications. Patients should consult healthcare providers before starting or stopping any other medications. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 65/100

Estradiol Transdermal received a safety concern score of 65/100 (elevated concern). This is based on a 49.8% serious event ratio across 41,509 classified reports. The score accounts for 79,078 total adverse event reports and 100 distinct reaction types. This elevated score indicates a notable proportion of serious adverse events and warrants careful monitoring.

Top Adverse Reactions

DRUG INEFFECTIVE3,429 reports
NAUSEA2,577 reports
FATIGUE2,572 reports
HEADACHE2,545 reports
OFF LABEL USE2,155 reports
PAIN1,870 reports
DIARRHOEA1,748 reports
BREAST CANCER FEMALE1,708 reports
DIZZINESS1,544 reports
ARTHRALGIA1,473 reports
PRODUCT ADHESION ISSUE1,425 reports
DYSPNOEA1,379 reports
RASH1,359 reports
PRURITUS1,331 reports
VOMITING1,223 reports
INSOMNIA1,219 reports
MALAISE1,143 reports
ANXIETY1,140 reports
HOT FLUSH1,108 reports
FEELING ABNORMAL1,042 reports
DEPRESSION1,012 reports
PRODUCT DOSE OMISSION ISSUE1,001 reports
PAIN IN EXTREMITY981 reports
ASTHENIA960 reports
WEIGHT INCREASED920 reports
FALL908 reports
DEVICE ADHESION ISSUE870 reports
CONDITION AGGRAVATED831 reports
BACK PAIN822 reports
WEIGHT DECREASED796 reports
COUGH795 reports
WRONG TECHNIQUE IN PRODUCT USAGE PROCESS781 reports
ALOPECIA765 reports
URINARY TRACT INFECTION728 reports
MUSCLE SPASMS727 reports
MIGRAINE719 reports
SINUSITIS702 reports
ABDOMINAL PAIN701 reports
HYPERSENSITIVITY681 reports
COVID 19675 reports
PRODUCT USE IN UNAPPROVED INDICATION674 reports
INJECTION SITE PAIN661 reports
PNEUMONIA661 reports
DRUG HYPERSENSITIVITY658 reports
CONSTIPATION655 reports
PARAESTHESIA644 reports
PRODUCT QUALITY ISSUE638 reports
HYPERTENSION629 reports
ABDOMINAL PAIN UPPER613 reports
BREAST CANCER607 reports
PYREXIA606 reports
ABDOMINAL DISCOMFORT602 reports
GAIT DISTURBANCE589 reports
URTICARIA583 reports
CHEST PAIN577 reports
DRUG INTERACTION575 reports
PRODUCT USE ISSUE573 reports
INCORRECT DOSE ADMINISTERED562 reports
HYPERHIDROSIS545 reports
HYPOAESTHESIA530 reports
NASOPHARYNGITIS530 reports
MYALGIA525 reports
PALPITATIONS515 reports
SOMNOLENCE508 reports
PERIPHERAL SWELLING495 reports
BLOOD PRESSURE INCREASED490 reports
MEMORY IMPAIRMENT490 reports
VISION BLURRED483 reports
TREMOR480 reports
ABDOMINAL DISTENSION478 reports
DECREASED APPETITE469 reports
ERYTHEMA460 reports
BRONCHITIS457 reports
CHRONIC KIDNEY DISEASE448 reports
INAPPROPRIATE SCHEDULE OF PRODUCT ADMINISTRATION439 reports
APPLICATION SITE ERYTHEMA431 reports
GASTROOESOPHAGEAL REFLUX DISEASE421 reports
PRODUCT SUBSTITUTION ISSUE409 reports
ASTHMA405 reports
APPLICATION SITE PRURITUS400 reports
JOINT SWELLING394 reports
NO ADVERSE EVENT393 reports
CONTUSION389 reports
CHEST DISCOMFORT381 reports
MUSCULAR WEAKNESS376 reports
DYSPEPSIA369 reports
OEDEMA PERIPHERAL368 reports
PSORIASIS368 reports
ACUTE KIDNEY INJURY364 reports
FLUSHING363 reports
ILLNESS361 reports
DEVICE ISSUE357 reports
EYE PAIN346 reports
BALANCE DISORDER341 reports
SUICIDAL IDEATION341 reports
OROPHARYNGEAL PAIN339 reports
VISUAL IMPAIRMENT339 reports
NIGHT SWEATS338 reports
SLEEP DISORDER336 reports
RHEUMATOID ARTHRITIS335 reports

Key Safety Signals

  • Breast cancer female (1708 reports)
  • Dizziness (1544 reports)
  • Drug interaction (575 reports)
  • Product quality issue (638 reports)
  • Product use issue (573 reports)

Patient Demographics

Adverse event reports by sex: Female: 38,052, Male: 724, Unknown: 86. The most frequently reported age groups are age 60 (829 reports), age 55 (825 reports), age 53 (806 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 41,509 classified reports for ESTRADIOL TRANSDERMAL:

  • Serious: 20,666 reports (49.8%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 20,843 reports (50.2%)
Serious 49.8%Non-Serious 50.2%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female38,052 (97.9%)
Male724 (1.9%)
Unknown86 (0.2%)

Reports by Age

Age 60829 reports
Age 55825 reports
Age 53806 reports
Age 54780 reports
Age 56759 reports
Age 58748 reports
Age 51744 reports
Age 57742 reports
Age 59742 reports
Age 52693 reports
Age 63676 reports
Age 61674 reports
Age 62651 reports
Age 50629 reports
Age 64607 reports
Age 65547 reports
Age 67538 reports
Age 69531 reports
Age 66530 reports
Age 68508 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Drug interactions are a key safety signal, with 575 reports indicating potential risks when combined with other medications. Patients should consult healthcare providers before starting or stopping any other medications.

What You Should Know

If you are taking Estradiol Transdermal, here are important things to know. The most commonly reported side effects include drug ineffective, nausea, fatigue, headache, off label use. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Follow prescribed usage instructions carefully to minimize the risk of adverse events. Report any unusual symptoms to your healthcare provider promptly. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA continues to monitor the safety of estradiol transdermal patches, and regulatory actions may be taken based on ongoing data analysis.

Frequently Asked Questions

How many adverse event reports has the FDA received for Estradiol Transdermal?

The FDA has received approximately 79,078 adverse event reports associated with Estradiol Transdermal. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Estradiol Transdermal?

The most frequently reported adverse events for Estradiol Transdermal include Drug Ineffective, Nausea, Fatigue, Headache, Off Label Use. By volume, the top reported reactions are: Drug Ineffective (3,429 reports), Nausea (2,577 reports), Fatigue (2,572 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Estradiol Transdermal.

What percentage of Estradiol Transdermal adverse event reports are serious?

Out of 41,509 classified reports, 20,666 (49.8%) were classified as serious and 20,843 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Estradiol Transdermal (by sex)?

Adverse event reports for Estradiol Transdermal break down by patient sex as follows: Female: 38,052, Male: 724, Unknown: 86. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Estradiol Transdermal?

The most frequently reported age groups for Estradiol Transdermal adverse events are: age 60: 829 reports, age 55: 825 reports, age 53: 806 reports, age 54: 780 reports, age 56: 759 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Estradiol Transdermal?

The primary manufacturer associated with Estradiol Transdermal adverse event reports is Amneal Pharmaceuticals Ny Llc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Estradiol Transdermal?

Beyond the most common reactions, other reported adverse events for Estradiol Transdermal include: Pain, Diarrhoea, Breast Cancer Female, Dizziness, Arthralgia. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Estradiol Transdermal?

You can report adverse events from Estradiol Transdermal to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Estradiol Transdermal's safety score and what does it mean?

Estradiol Transdermal has a safety concern score of 65 out of 100 (elevated concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. The most common reactions include nausea, fatigue, and headache, indicating a broad range of mild to moderate side effects.

What are the key safety signals for Estradiol Transdermal?

Key safety signals identified in Estradiol Transdermal's adverse event data include: Breast cancer female (1708 reports). Dizziness (1544 reports). Drug interaction (575 reports). Product quality issue (638 reports). Product use issue (573 reports). These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Estradiol Transdermal interact with other drugs?

Drug interactions are a key safety signal, with 575 reports indicating potential risks when combined with other medications. Patients should consult healthcare providers before starting or stopping any other medications. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Estradiol Transdermal.

What should patients know before taking Estradiol Transdermal?

Follow prescribed usage instructions carefully to minimize the risk of adverse events. Report any unusual symptoms to your healthcare provider promptly.

Are Estradiol Transdermal side effects well-documented?

Estradiol Transdermal has 79,078 adverse event reports on file with the FDA. Serious adverse events, such as breast cancer and dizziness, are reported but at a lower frequency compared to non-serious events. The volume of reports for Estradiol Transdermal reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Estradiol Transdermal?

The FDA continues to monitor the safety of estradiol transdermal patches, and regulatory actions may be taken based on ongoing data analysis. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to ESTRADIOL TRANSDERMAL based on therapeutic use, drug class, or shared indications:

IbuprofenMetforminWarfarin
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.