TOFACITINIB

72/100 · Elevated

Manufactured by Pfizer Laboratories Div Pfizer Inc

Tofacitinib Adverse Events: Pain and Fatigue Predominate, with Serious Reactions Notably High

696,662 FDA adverse event reports analyzed

Last updated: 2026-05-12

About TOFACITINIB

TOFACITINIB is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Pfizer Laboratories Div Pfizer Inc. Based on analysis of 696,662 FDA adverse event reports, TOFACITINIB has a safety score of 72 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for TOFACITINIB include DRUG INEFFECTIVE, PAIN, ARTHRALGIA, CONDITION AGGRAVATED, RHEUMATOID ARTHRITIS. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for TOFACITINIB.

AI Safety Analysis

Tofacitinib has a safety concern score of 72 out of 100, placing it in the elevated concern category based on analysis of FDA adverse event data. The FDA has received approximately 696,662 adverse event reports for this medication, which is primarily manufactured by Pfizer Laboratories Div Pfizer Inc.

The most commonly reported adverse events include Drug Ineffective, Pain, Arthralgia. Of classified reports, 47.7% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Pain and fatigue are the most common adverse reactions, with over 25,000 reports each.

Serious adverse events account for nearly half of all reports, indicating significant safety concerns. The reaction diversity is high, with over 100 distinct reactions reported.

Patients taking Tofacitinib should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Tofacitinib can cause serious infections and liver enzyme increases, and patients should be monitored for these conditions. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 72/100

Tofacitinib received a safety concern score of 72/100 (elevated concern). This is based on a 47.7% serious event ratio across 181,992 classified reports. The score accounts for 696,662 total adverse event reports and 100 distinct reaction types. This elevated score indicates a notable proportion of serious adverse events and warrants careful monitoring.

Top Adverse Reactions

DRUG INEFFECTIVE43,542 reports
PAIN25,737 reports
ARTHRALGIA19,670 reports
CONDITION AGGRAVATED19,467 reports
RHEUMATOID ARTHRITIS18,797 reports
FATIGUE16,595 reports
OFF LABEL USE14,815 reports
JOINT SWELLING14,455 reports
HEADACHE13,405 reports
RASH11,912 reports
DRUG INTOLERANCE11,718 reports
MALAISE10,489 reports
PAIN IN EXTREMITY10,277 reports
ABDOMINAL DISCOMFORT10,168 reports
NAUSEA9,949 reports
DIARRHOEA9,695 reports
PERIPHERAL SWELLING9,668 reports
ALOPECIA9,255 reports
MUSCULOSKELETAL STIFFNESS9,233 reports
SYNOVITIS9,206 reports
SWELLING9,194 reports
ARTHROPATHY9,131 reports
NASOPHARYNGITIS8,699 reports
TREATMENT FAILURE8,527 reports
DRUG HYPERSENSITIVITY8,362 reports
CONTRAINDICATED PRODUCT ADMINISTERED8,286 reports
HYPERSENSITIVITY7,906 reports
INFECTION7,678 reports
HEPATIC ENZYME INCREASED7,657 reports
SYSTEMIC LUPUS ERYTHEMATOSUS6,894 reports
HAND DEFORMITY6,863 reports
THERAPEUTIC PRODUCT EFFECT DECREASED6,738 reports
INFUSION RELATED REACTION6,436 reports
DYSPNOEA6,331 reports
GLOSSODYNIA6,230 reports
PEMPHIGUS6,204 reports
PNEUMONIA6,201 reports
THERAPEUTIC PRODUCT EFFECT INCOMPLETE6,197 reports
WEIGHT INCREASED6,197 reports
SINUSITIS6,121 reports
HYPERTENSION6,111 reports
PRODUCT USE ISSUE6,016 reports
WOUND5,962 reports
PRODUCT DOSE OMISSION ISSUE5,825 reports
PYREXIA5,712 reports
BLOOD CHOLESTEROL INCREASED5,677 reports
VOMITING5,382 reports
DISCOMFORT5,367 reports
PERICARDITIS5,274 reports
COVID 195,266 reports
ANTI CYCLIC CITRULLINATED PEPTIDE ANTIBODY POSITIVE5,124 reports
MOBILITY DECREASED5,040 reports
DIZZINESS4,862 reports
PRURITUS4,858 reports
ABDOMINAL PAIN UPPER4,854 reports
GAIT DISTURBANCE4,772 reports
FALL4,448 reports
ARTHRITIS4,433 reports
GASTROINTESTINAL DISORDER4,421 reports
LOSS OF PERSONAL INDEPENDENCE IN DAILY ACTIVITIES4,391 reports
MATERNAL EXPOSURE DURING PREGNANCY4,388 reports
HELICOBACTER INFECTION4,343 reports
INFLAMMATION4,260 reports
STOMATITIS4,219 reports
GENERAL PHYSICAL HEALTH DETERIORATION4,211 reports
CONFUSIONAL STATE4,173 reports
COUGH4,161 reports
MEMORY IMPAIRMENT4,158 reports
IMPAIRED HEALING4,129 reports
DUODENAL ULCER PERFORATION4,120 reports
ILLNESS4,111 reports
HERPES ZOSTER4,083 reports
INSOMNIA4,074 reports
BLISTER4,061 reports
HYPOAESTHESIA4,054 reports
ASTHENIA4,036 reports
RHEUMATOID FACTOR POSITIVE3,825 reports
LOWER RESPIRATORY TRACT INFECTION3,786 reports
PSORIATIC ARTHROPATHY3,772 reports
BACK PAIN3,770 reports
DEPRESSION3,711 reports
OSTEOARTHRITIS3,666 reports
INTENTIONAL PRODUCT USE ISSUE3,656 reports
FIBROMYALGIA3,634 reports
IRRITABLE BOWEL SYNDROME3,595 reports
CONTUSION3,580 reports
DEATH3,523 reports
URINARY TRACT INFECTION3,518 reports
URTICARIA3,467 reports
FOLLICULITIS3,465 reports
C REACTIVE PROTEIN INCREASED3,357 reports
PRODUCT USE IN UNAPPROVED INDICATION3,270 reports
TYPE 2 DIABETES MELLITUS3,227 reports
MUSCULOSKELETAL PAIN3,208 reports
ILL DEFINED DISORDER3,129 reports
C REACTIVE PROTEIN ABNORMAL3,116 reports
MUSCLE INJURY3,102 reports
SLEEP DISORDER3,069 reports
MUSCLE SPASMS2,974 reports
INFLUENZA2,961 reports

Key Safety Signals

  • Pain and arthralgia are the most frequently reported conditions, suggesting potential musculoskeletal issues.
  • Serious infections, including pneumonia and sepsis, are notable, with over 7,600 reports.
  • Liver enzyme increases and systemic lupus erythematosus are also significant safety signals.

Patient Demographics

Adverse event reports by sex: Female: 138,558, Male: 33,777, Unknown: 277. The most frequently reported age groups are age 63 (4,935 reports), age 61 (4,791 reports), age 60 (4,788 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 181,992 classified reports for TOFACITINIB:

  • Serious: 86,746 reports (47.7%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 95,246 reports (52.3%)
Serious 47.7%Non-Serious 52.3%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female138,558 (80.3%)
Male33,777 (19.6%)
Unknown277 (0.2%)

Reports by Age

Age 634,935 reports
Age 614,791 reports
Age 604,788 reports
Age 654,668 reports
Age 594,654 reports
Age 644,577 reports
Age 624,543 reports
Age 584,499 reports
Age 574,074 reports
Age 564,026 reports
Age 674,020 reports
Age 663,907 reports
Age 683,750 reports
Age 553,730 reports
Age 543,698 reports
Age 693,591 reports
Age 703,512 reports
Age 443,463 reports
Age 533,305 reports
Age 713,261 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Tofacitinib can cause serious infections and liver enzyme increases, and patients should be monitored for these conditions.

What You Should Know

If you are taking Tofacitinib, here are important things to know. The most commonly reported side effects include drug ineffective, pain, arthralgia, condition aggravated, rheumatoid arthritis. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Patients should report any new or worsening symptoms to their healthcare provider immediately. Regular monitoring of liver function and infection risk is recommended. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA continues to monitor the safety of tofacitinib, and updates will be provided as necessary based on ongoing studies.

Frequently Asked Questions

How many adverse event reports has the FDA received for Tofacitinib?

The FDA has received approximately 696,662 adverse event reports associated with Tofacitinib. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Tofacitinib?

The most frequently reported adverse events for Tofacitinib include Drug Ineffective, Pain, Arthralgia, Condition Aggravated, Rheumatoid Arthritis. By volume, the top reported reactions are: Drug Ineffective (43,542 reports), Pain (25,737 reports), Arthralgia (19,670 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Tofacitinib.

What percentage of Tofacitinib adverse event reports are serious?

Out of 181,992 classified reports, 86,746 (47.7%) were classified as serious and 95,246 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Tofacitinib (by sex)?

Adverse event reports for Tofacitinib break down by patient sex as follows: Female: 138,558, Male: 33,777, Unknown: 277. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Tofacitinib?

The most frequently reported age groups for Tofacitinib adverse events are: age 63: 4,935 reports, age 61: 4,791 reports, age 60: 4,788 reports, age 65: 4,668 reports, age 59: 4,654 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Tofacitinib?

The primary manufacturer associated with Tofacitinib adverse event reports is Pfizer Laboratories Div Pfizer Inc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Tofacitinib?

Beyond the most common reactions, other reported adverse events for Tofacitinib include: Fatigue, Off Label Use, Joint Swelling, Headache, Rash. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Tofacitinib?

You can report adverse events from Tofacitinib to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Tofacitinib's safety score and what does it mean?

Tofacitinib has a safety concern score of 72 out of 100 (elevated concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Pain and fatigue are the most common adverse reactions, with over 25,000 reports each.

What are the key safety signals for Tofacitinib?

Key safety signals identified in Tofacitinib's adverse event data include: Pain and arthralgia are the most frequently reported conditions, suggesting potential musculoskeletal issues.. Serious infections, including pneumonia and sepsis, are notable, with over 7,600 reports.. Liver enzyme increases and systemic lupus erythematosus are also significant safety signals.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Tofacitinib interact with other drugs?

Tofacitinib can cause serious infections and liver enzyme increases, and patients should be monitored for these conditions. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Tofacitinib.

What should patients know before taking Tofacitinib?

Patients should report any new or worsening symptoms to their healthcare provider immediately. Regular monitoring of liver function and infection risk is recommended.

Are Tofacitinib side effects well-documented?

Tofacitinib has 696,662 adverse event reports on file with the FDA. Serious adverse events account for nearly half of all reports, indicating significant safety concerns. The volume of reports for Tofacitinib reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Tofacitinib?

The FDA continues to monitor the safety of tofacitinib, and updates will be provided as necessary based on ongoing studies. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to TOFACITINIB based on therapeutic use, drug class, or shared indications:

AbacavirRitonavirCobicistat
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.