VARENICLINE TARTRATE

85/100 · Critical

Manufactured by Pfizer Laboratories Div Pfizer Inc

High Safety Concerns with Varenicline Tartrate, Particularly for Mental Health and Suicide-Related Reactions

167,559 FDA adverse event reports analyzed

Last updated: 2026-05-12

About VARENICLINE TARTRATE

VARENICLINE TARTRATE is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Pfizer Laboratories Div Pfizer Inc. Based on analysis of 167,559 FDA adverse event reports, VARENICLINE TARTRATE has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for VARENICLINE TARTRATE include NAUSEA, DEPRESSION, ABNORMAL DREAMS, ANXIETY, DRUG INEFFECTIVE. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for VARENICLINE TARTRATE.

AI Safety Analysis

Varenicline Tartrate has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 167,559 adverse event reports for this medication, which is primarily manufactured by Pfizer Laboratories Div Pfizer Inc.

The most commonly reported adverse events include Nausea, Depression, Abnormal Dreams. Of classified reports, 40.6% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. Significant reports of depression, suicidal ideation, and suicide attempts, indicating potential mental health risks.

Nausea and vomiting are common gastrointestinal side effects. Drug interactions and intolerances are reported, necessitating careful monitoring. Serious adverse events, including chest pain and myocardial infarction, are notable but less frequent. Weight changes and mood swings are also commonly reported.

Patients taking Varenicline Tartrate should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Varenicline Tartrate can interact with other drugs, and patients should be monitored for adverse reactions. Patients with a history of mental health issues should be closely observed. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Varenicline Tartrate received a safety concern score of 85/100 (high concern). This is based on a 40.6% serious event ratio across 79,201 classified reports. The score accounts for 167,559 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

NAUSEA14,427 reports
DEPRESSION8,667 reports
ABNORMAL DREAMS7,824 reports
ANXIETY5,940 reports
DRUG INEFFECTIVE5,640 reports
INSOMNIA5,566 reports
VOMITING4,581 reports
SUICIDAL IDEATION4,194 reports
HEADACHE4,139 reports
FEELING ABNORMAL3,989 reports
MALAISE3,982 reports
NIGHTMARE3,349 reports
FATIGUE3,163 reports
DIZZINESS3,018 reports
AGGRESSION2,772 reports
SUICIDE ATTEMPT2,253 reports
ANGER2,250 reports
IRRITABILITY2,229 reports
CONSTIPATION2,208 reports
AGITATION2,092 reports
DYSPNOEA2,071 reports
WEIGHT INCREASED1,976 reports
ABDOMINAL DISCOMFORT1,854 reports
ABDOMINAL PAIN UPPER1,812 reports
SOMNOLENCE1,786 reports
DIARRHOEA1,770 reports
ABNORMAL BEHAVIOUR1,669 reports
FLATULENCE1,666 reports
RASH1,597 reports
PAIN1,593 reports
DYSGEUSIA1,590 reports
SLEEP DISORDER1,522 reports
MENTAL DISORDER1,507 reports
WEIGHT DECREASED1,466 reports
NERVOUSNESS1,431 reports
MOOD SWINGS1,349 reports
DRUG INTERACTION1,182 reports
STRESS1,161 reports
ASTHENIA1,133 reports
PRURITUS1,131 reports
CHEST PAIN1,129 reports
TREMOR1,125 reports
LOSS OF CONSCIOUSNESS1,076 reports
DEPRESSED MOOD1,057 reports
MEMORY IMPAIRMENT1,034 reports
HALLUCINATION1,017 reports
CRYING1,003 reports
INTENTIONAL OVERDOSE994 reports
DECREASED APPETITE987 reports
DRUG HYPERSENSITIVITY975 reports
MOOD ALTERED961 reports
CONFUSIONAL STATE931 reports
AMNESIA919 reports
PANIC ATTACK907 reports
ARTHRALGIA889 reports
DISTURBANCE IN ATTENTION882 reports
ABDOMINAL DISTENSION858 reports
PARANOIA848 reports
COUGH807 reports
BACK PAIN795 reports
PALPITATIONS794 reports
TOBACCO USER793 reports
COMPLETED SUICIDE784 reports
FALL784 reports
HYPERTENSION783 reports
THINKING ABNORMAL765 reports
EMOTIONAL DISORDER758 reports
MUSCLE SPASMS749 reports
PAIN IN EXTREMITY726 reports
CHRONIC OBSTRUCTIVE PULMONARY DISEASE723 reports
HYPERSENSITIVITY714 reports
CONVULSION698 reports
HYPERHIDROSIS691 reports
DYSPEPSIA690 reports
BLOOD PRESSURE INCREASED681 reports
VISION BLURRED668 reports
ABDOMINAL PAIN641 reports
MYALGIA627 reports
PSYCHOTIC DISORDER604 reports
MYOCARDIAL INFARCTION591 reports
PNEUMONIA591 reports
BLOOD GLUCOSE INCREASED587 reports
URTICARIA579 reports
HOMICIDAL IDEATION558 reports
EMOTIONAL DISTRESS553 reports
INCORRECT DOSE ADMINISTERED547 reports
HYPOAESTHESIA546 reports
DRUG INTOLERANCE533 reports
CONDITION AGGRAVATED531 reports
PARAESTHESIA530 reports
BIPOLAR DISORDER527 reports
GAIT DISTURBANCE511 reports
THERAPEUTIC RESPONSE UNEXPECTED508 reports
PERSONALITY CHANGE503 reports
DRY MOUTH501 reports
HEART RATE INCREASED495 reports
MIGRAINE494 reports
ACTIVITIES OF DAILY LIVING IMPAIRED493 reports
CEREBROVASCULAR ACCIDENT492 reports
DRUG DOSE OMISSION473 reports

Key Safety Signals

  • Suicidal ideation and suicide attempts
  • Depression and depressive mood
  • Drug interactions and intolerances

Patient Demographics

Adverse event reports by sex: Female: 45,796, Male: 25,889, Unknown: 427. The most frequently reported age groups are age 58 (809 reports), age 55 (792 reports), age 60 (761 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 79,201 classified reports for VARENICLINE TARTRATE:

  • Serious: 32,170 reports (40.6%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 47,031 reports (59.4%)
Serious 40.6%Non-Serious 59.4%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Female45,796 (63.5%)
Male25,889 (35.9%)
Unknown427 (0.6%)

Reports by Age

Age 58809 reports
Age 55792 reports
Age 60761 reports
Age 53758 reports
Age 52746 reports
Age 50718 reports
Age 57706 reports
Age 56704 reports
Age 61692 reports
Age 54691 reports
Age 59690 reports
Age 62681 reports
Age 63681 reports
Age 51648 reports
Age 48587 reports
Age 64587 reports
Age 65553 reports
Age 49543 reports
Age 47537 reports
Age 45524 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Varenicline Tartrate can interact with other drugs, and patients should be monitored for adverse reactions. Patients with a history of mental health issues should be closely observed.

What You Should Know

If you are taking Varenicline Tartrate, here are important things to know. The most commonly reported side effects include nausea, depression, abnormal dreams, anxiety, drug ineffective. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Patients should report any new or worsening mental health symptoms to their healthcare provider immediately. Follow prescribed dosing instructions carefully to avoid drug interactions and intolerances. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

The FDA has issued warnings about the potential for serious mental health effects, including suicidal ideation and depression. Healthcare providers should be vigilant and consider alternative treatments for patients with a history of mental health is

Frequently Asked Questions

How many adverse event reports has the FDA received for Varenicline Tartrate?

The FDA has received approximately 167,559 adverse event reports associated with Varenicline Tartrate. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Varenicline Tartrate?

The most frequently reported adverse events for Varenicline Tartrate include Nausea, Depression, Abnormal Dreams, Anxiety, Drug Ineffective. By volume, the top reported reactions are: Nausea (14,427 reports), Depression (8,667 reports), Abnormal Dreams (7,824 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Varenicline Tartrate.

What percentage of Varenicline Tartrate adverse event reports are serious?

Out of 79,201 classified reports, 32,170 (40.6%) were classified as serious and 47,031 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Varenicline Tartrate (by sex)?

Adverse event reports for Varenicline Tartrate break down by patient sex as follows: Female: 45,796, Male: 25,889, Unknown: 427. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Varenicline Tartrate?

The most frequently reported age groups for Varenicline Tartrate adverse events are: age 58: 809 reports, age 55: 792 reports, age 60: 761 reports, age 53: 758 reports, age 52: 746 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Varenicline Tartrate?

The primary manufacturer associated with Varenicline Tartrate adverse event reports is Pfizer Laboratories Div Pfizer Inc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Varenicline Tartrate?

Beyond the most common reactions, other reported adverse events for Varenicline Tartrate include: Insomnia, Vomiting, Suicidal Ideation, Headache, Feeling Abnormal. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Varenicline Tartrate?

You can report adverse events from Varenicline Tartrate to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Varenicline Tartrate's safety score and what does it mean?

Varenicline Tartrate has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. Significant reports of depression, suicidal ideation, and suicide attempts, indicating potential mental health risks.

What are the key safety signals for Varenicline Tartrate?

Key safety signals identified in Varenicline Tartrate's adverse event data include: Suicidal ideation and suicide attempts. Depression and depressive mood. Drug interactions and intolerances. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Varenicline Tartrate interact with other drugs?

Varenicline Tartrate can interact with other drugs, and patients should be monitored for adverse reactions. Patients with a history of mental health issues should be closely observed. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Varenicline Tartrate.

What should patients know before taking Varenicline Tartrate?

Patients should report any new or worsening mental health symptoms to their healthcare provider immediately. Follow prescribed dosing instructions carefully to avoid drug interactions and intolerances.

Are Varenicline Tartrate side effects well-documented?

Varenicline Tartrate has 167,559 adverse event reports on file with the FDA. Nausea and vomiting are common gastrointestinal side effects. The volume of reports for Varenicline Tartrate reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Varenicline Tartrate?

The FDA has issued warnings about the potential for serious mental health effects, including suicidal ideation and depression. Healthcare providers should be vigilant and consider alternative treatments for patients with a history of mental health is For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to VARENICLINE TARTRATE based on therapeutic use, drug class, or shared indications:

ParoxetineSertralineFluoxetineEscitalopramBupropion
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.