TEMOZOLOMIDE

85/100 · Critical

Manufactured by Merck Sharp & Dohme LLC

High Safety Concerns with Temozolomide, Particularly for Serious Adverse Events

38,373 FDA adverse event reports analyzed

Last updated: 2026-05-12

About TEMOZOLOMIDE

TEMOZOLOMIDE is a medication tracked in the FDA Adverse Event Reporting System (FAERS), manufactured by Merck Sharp & Dohme LLC. Based on analysis of 38,373 FDA adverse event reports, TEMOZOLOMIDE has a safety score of 85 out of 100. This score indicates a relatively favorable safety profile, with fewer or less severe adverse events compared to many other tracked medications. The most commonly reported adverse reactions for TEMOZOLOMIDE include DISEASE PROGRESSION, DEATH, OFF LABEL USE, THROMBOCYTOPENIA, PRODUCT USE IN UNAPPROVED INDICATION. This page provides a comprehensive breakdown of reported side effects, safety signals, patient demographics, and AI-powered safety analysis for TEMOZOLOMIDE.

AI Safety Analysis

Temozolomide has a safety concern score of 85 out of 100, placing it in the high concern category based on analysis of FDA adverse event data. The FDA has received approximately 38,373 adverse event reports for this medication, which is primarily manufactured by Merck Sharp & Dohme Llc.

The most commonly reported adverse events include Disease Progression, Death, Off Label Use. Of classified reports, 81.0% were designated as serious by the FDA, meaning they involved hospitalization, disability, or other significant medical outcomes. High incidence of serious adverse events such as disease progression and death.

Significant hematological toxicity, including thrombocytopenia and neutropenia. Common gastrointestinal issues like nausea and vomiting.

Patients taking Temozolomide should monitor for the commonly reported side effects and contact their healthcare provider if they experience any unusual symptoms. Temozolomide can cause severe hematological and gastrointestinal side effects, and patients should be monitored closely for these issues. Drug interactions, particularly with other hematological agents, should be carefully managed. This analysis is based on voluntary FDA adverse event reports and should not replace professional medical advice.

Safety Score: 85/100

Temozolomide received a safety concern score of 85/100 (high concern). This is based on a 81.0% serious event ratio across 20,264 classified reports. The score accounts for 38,373 total adverse event reports and 100 distinct reaction types. This high score reflects a significant proportion of serious adverse events in the reporting data.

Top Adverse Reactions

DISEASE PROGRESSION1,849 reports
DEATH1,683 reports
OFF LABEL USE1,640 reports
THROMBOCYTOPENIA1,519 reports
PRODUCT USE IN UNAPPROVED INDICATION1,390 reports
NAUSEA1,264 reports
DRUG INEFFECTIVE1,232 reports
FATIGUE1,007 reports
NEUTROPENIA1,001 reports
VOMITING948 reports
MALIGNANT NEOPLASM PROGRESSION889 reports
FEBRILE NEUTROPENIA813 reports
DIARRHOEA753 reports
ANAEMIA723 reports
ASTHENIA631 reports
PLATELET COUNT DECREASED615 reports
PYREXIA614 reports
INFECTION559 reports
HEADACHE548 reports
PANCYTOPENIA496 reports
CONSTIPATION452 reports
SEIZURE451 reports
NEOPLASM PROGRESSION432 reports
PULMONARY EMBOLISM417 reports
PNEUMONIA415 reports
HAEMORRHAGE400 reports
ATRIAL FIBRILLATION375 reports
CONFUSIONAL STATE372 reports
CYTOPENIA353 reports
LYMPHOPENIA350 reports
DEHYDRATION341 reports
FALL339 reports
SEPSIS339 reports
DYSPNOEA337 reports
DECREASED APPETITE331 reports
WHITE BLOOD CELL COUNT DECREASED328 reports
ASPERGILLUS INFECTION327 reports
CONVULSION324 reports
DISEASE RECURRENCE315 reports
MYELOSUPPRESSION310 reports
WEIGHT DECREASED297 reports
LEUKOPENIA295 reports
RASH289 reports
PAIN287 reports
ABDOMINAL PAIN283 reports
BONE MARROW FAILURE277 reports
DEEP VEIN THROMBOSIS271 reports
TOXICITY TO VARIOUS AGENTS246 reports
GLIOBLASTOMA241 reports
METASTASES TO LIVER236 reports
HYPERTENSION231 reports
PRODUCT USE ISSUE224 reports
HAEMATOTOXICITY223 reports
HYPOTENSION222 reports
HAEMOGLOBIN DECREASED210 reports
DIZZINESS205 reports
ALANINE AMINOTRANSFERASE INCREASED199 reports
GAIT DISTURBANCE199 reports
HOSPITALISATION196 reports
BRAIN OEDEMA190 reports
ACUTE KIDNEY INJURY189 reports
THERAPY PARTIAL RESPONDER189 reports
GENERAL PHYSICAL HEALTH DETERIORATION188 reports
MUSCULAR WEAKNESS188 reports
MENTAL STATUS CHANGES187 reports
NEUTROPHIL COUNT DECREASED187 reports
URINARY TRACT INFECTION186 reports
MALAISE183 reports
SOMNOLENCE183 reports
TUMOUR PSEUDOPROGRESSION182 reports
DRUG INTERACTION173 reports
HEMIPARESIS172 reports
HOSPICE CARE170 reports
CONDITION AGGRAVATED165 reports
HYPONATRAEMIA162 reports
COUGH160 reports
GLIOBLASTOMA MULTIFORME154 reports
HYPERGLYCAEMIA153 reports
PAIN IN EXTREMITY153 reports
HYPOKALAEMIA148 reports
DYSPHAGIA146 reports
APLASTIC ANAEMIA144 reports
LYMPHOCYTE COUNT DECREASED144 reports
CHILLS143 reports
ARTHRALGIA142 reports
APHASIA141 reports
ASPARTATE AMINOTRANSFERASE INCREASED140 reports
HYPERMUTATION132 reports
RESPIRATORY FAILURE130 reports
BACK PAIN129 reports
COGNITIVE DISORDER129 reports
CHEST PAIN128 reports
LETHARGY127 reports
OEDEMA PERIPHERAL125 reports
THROMBOSIS118 reports
EPISTAXIS117 reports
SEPTIC SHOCK117 reports
MUCOSAL INFLAMMATION116 reports
DRUG RESISTANCE115 reports
METASTASES TO CENTRAL NERVOUS SYSTEM115 reports

Key Safety Signals

  • High number of reports of disease progression and death.
  • Severe hematological effects including thrombocytopenia and neutropenia.
  • Frequent gastrointestinal side effects such as nausea and vomiting.

Patient Demographics

Adverse event reports by sex: Male: 9,249, Female: 7,868, Unknown: 171. The most frequently reported age groups are age 59 (343 reports), age 67 (323 reports), age 65 (316 reports). These demographics reflect reporting patterns and may not represent the full patient population.

Report Outcomes

Out of 20,264 classified reports for TEMOZOLOMIDE:

  • Serious: 16,404 reports (81.0%) — includes hospitalization, disability, life-threatening events, or death
  • Non-Serious: 3,860 reports (19.0%)
Serious 81.0%Non-Serious 19.0%

The FDA classifies an adverse event as “serious” if it results in death, hospitalization, disability, congenital anomaly, or requires intervention to prevent permanent damage.

Demographics Breakdown

Reports by Sex

Male9,249 (53.5%)
Female7,868 (45.5%)
Unknown171 (1.0%)

Reports by Age

Age 59343 reports
Age 67323 reports
Age 65316 reports
Age 66316 reports
Age 64314 reports
Age 61304 reports
Age 62301 reports
Age 58299 reports
Age 69297 reports
Age 55293 reports
Age 68293 reports
Age 63279 reports
Age 57278 reports
Age 60274 reports
Age 53271 reports
Age 71257 reports
Age 56251 reports
Age 54245 reports
Age 50243 reports
Age 70240 reports

Demographics reflect voluntary FDA adverse event reporting patterns and may not represent the full patient population.

Drug Interactions & Warnings

Temozolomide can cause severe hematological and gastrointestinal side effects, and patients should be monitored closely for these issues. Drug interactions, particularly with other hematological agents, should be carefully managed.

What You Should Know

If you are taking Temozolomide, here are important things to know. The most commonly reported side effects include disease progression, death, off label use, thrombocytopenia, product use in unapproved indication. While many of these may be mild and temporary, you should contact your healthcare provider if any symptoms are severe or persistent. Monitor patients closely for signs of hematological toxicity and gastrointestinal issues. Be aware of potential drug interactions, especially with other hematological agents. If you experience a serious adverse reaction, seek emergency medical attention immediately or call 911. You can report side effects to the FDA's MedWatch program at 1-800-FDA-1088.

Regulatory Context

Regulatory oversight is ongoing, with a focus on monitoring hematological and gastrointestinal toxicity. Healthcare providers should report any adverse events to the FDA.

Frequently Asked Questions

How many adverse event reports has the FDA received for Temozolomide?

The FDA has received approximately 38,373 adverse event reports associated with Temozolomide. These reports come from healthcare professionals, consumers, and manufacturers through the FDA Adverse Event Reporting System (FAERS). Note that the number of reports does not directly indicate the frequency of side effects, as adverse events are voluntarily reported and may be underrepresented.

What are the most commonly reported side effects of Temozolomide?

The most frequently reported adverse events for Temozolomide include Disease Progression, Death, Off Label Use, Thrombocytopenia, Product Use In Unapproved Indication. By volume, the top reported reactions are: Disease Progression (1,849 reports), Death (1,683 reports), Off Label Use (1,640 reports). These figures reflect FDA adverse event reports and may not represent the true incidence rate of these side effects in all patients taking Temozolomide.

What percentage of Temozolomide adverse event reports are serious?

Out of 20,264 classified reports, 16,404 (81.0%) were classified as serious and 3,860 as non-serious. The FDA classifies an event as "serious" if it results in death, hospitalization, disability, or other medically significant outcomes. A higher serious-event ratio warrants closer attention but does not necessarily mean the drug is unsafe.

Who reports adverse events for Temozolomide (by sex)?

Adverse event reports for Temozolomide break down by patient sex as follows: Male: 9,249, Female: 7,868, Unknown: 171. This distribution reflects reporting patterns rather than actual risk differences between groups. Reporting rates can be influenced by prescribing patterns, disease demographics, and reporting behavior.

What age groups report the most side effects for Temozolomide?

The most frequently reported age groups for Temozolomide adverse events are: age 59: 343 reports, age 67: 323 reports, age 65: 316 reports, age 66: 316 reports, age 64: 314 reports. Age-related reporting patterns can reflect both the demographics of the patient population and potential age-related susceptibility to certain side effects.

Who manufactures Temozolomide?

The primary manufacturer associated with Temozolomide adverse event reports is Merck Sharp & Dohme Llc. Multiple manufacturers may produce generic versions of this drug. The manufacturer listed reflects the most frequently reported brand in FDA adverse event data.

What other side effects have been reported for Temozolomide?

Beyond the most common reactions, other reported adverse events for Temozolomide include: Nausea, Drug Ineffective, Fatigue, Neutropenia, Vomiting. Less common side effects can still be clinically significant. Patients should report any unusual symptoms to their healthcare provider.

How do I report a side effect from Temozolomide?

You can report adverse events from Temozolomide to the FDA through their MedWatch program at www.fda.gov/medwatch, by calling 1-800-FDA-1088, or by completing Form FDA 3500. Healthcare professionals, consumers, and manufacturers can all submit reports. Reporting helps the FDA monitor drug safety after approval.

What is Temozolomide's safety score and what does it mean?

Temozolomide has a safety concern score of 85 out of 100 (high concern). This score is calculated from the ratio of serious to non-serious adverse events, the diversity of reported reactions, and the overall volume of reports relative to usage. High incidence of serious adverse events such as disease progression and death.

What are the key safety signals for Temozolomide?

Key safety signals identified in Temozolomide's adverse event data include: High number of reports of disease progression and death.. Severe hematological effects including thrombocytopenia and neutropenia.. Frequent gastrointestinal side effects such as nausea and vomiting.. These signals are derived from patterns in FDA reports and should be discussed with a healthcare provider for personalized assessment.

Does Temozolomide interact with other drugs?

Temozolomide can cause severe hematological and gastrointestinal side effects, and patients should be monitored closely for these issues. Drug interactions, particularly with other hematological agents, should be carefully managed. Always inform your healthcare provider about all medications, supplements, and over-the-counter drugs you are taking before starting Temozolomide.

What should patients know before taking Temozolomide?

Monitor patients closely for signs of hematological toxicity and gastrointestinal issues. Be aware of potential drug interactions, especially with other hematological agents.

Are Temozolomide side effects well-documented?

Temozolomide has 38,373 adverse event reports on file with the FDA. Significant hematological toxicity, including thrombocytopenia and neutropenia. The volume of reports for Temozolomide reflects both the drug's usage level and the vigilance of the reporting community.

What is the FDA's position on Temozolomide?

Regulatory oversight is ongoing, with a focus on monitoring hematological and gastrointestinal toxicity. Healthcare providers should report any adverse events to the FDA. For the most current regulatory information, check the FDA's drug labeling database or consult your pharmacist.

Related Drugs

Drugs related to TEMOZOLOMIDE based on therapeutic use, drug class, or shared indications:

CyclophosphamideVincristineFludarabine
Important Disclaimer: This content is generated by AI analysis of FDA adverse event reports and is provided for informational purposes only. It is not medical advice. Adverse event reports submitted to the FDA do not prove that a medication caused the reported side effect. Always consult your healthcare provider before starting, stopping, or changing any medication. If you experience a serious side effect, contact your doctor or call 911 immediately.